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Found 11 of ic50 for monomerid = 50005410
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Jilin University

Curated by ChEMBL
LigandPNGBDBM50005410(CHEMBL139197 | CHEMBL2137199)
Affinity DataIC50:  110nMAssay Description:Inhibition of Gal4-RORgamma-LBD (180 to 507 residues) (unknown origin) expressed in HEK293T cells after 24 hrs by dual-luciferase reporter assayMore data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Jilin University

Curated by ChEMBL
LigandPNGBDBM50005410(CHEMBL139197 | CHEMBL2137199)
Affinity DataIC50:  150nMAssay Description:Displacement of [3H]T0901317 from human RoRc expressed in HepG2 cells by scintillation proximity binding assayMore data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Jilin University

Curated by ChEMBL
LigandPNGBDBM50005410(CHEMBL139197 | CHEMBL2137199)
Affinity DataIC50:  320nMAssay Description:Inhibition of human GAL4-fused RORgamma transfected in HEK293 cells co-transfected with G6Pase by luciferase reporter assayMore data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Jilin University

Curated by ChEMBL
LigandPNGBDBM50005410(CHEMBL139197 | CHEMBL2137199)
Affinity DataIC50:  420nMAssay Description:Antagonist activity at full-length RORgamma (unknown origin) expressed in 293T cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Jilin University

Curated by ChEMBL
LigandPNGBDBM50005410(CHEMBL139197 | CHEMBL2137199)
Affinity DataIC50:  430nMAssay Description:Antagonist activity at Gal4-fused RORgamma (unknown origin) expressed in 293T cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Jilin University

Curated by ChEMBL
LigandPNGBDBM50005410(CHEMBL139197 | CHEMBL2137199)
Affinity DataIC50:  910nMAssay Description:Displacement of N-terminal biotinylated SRC1-4 coactivator peptide from N-terminal His6-fused human RORgamma-LBD (262 to 507 residues) expressed in E...More data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Jilin University

Curated by ChEMBL
LigandPNGBDBM50005410(CHEMBL139197 | CHEMBL2137199)
Affinity DataIC50:  3.54E+3nMAssay Description:Antagonist activity at human His6-tagged RORgamma ligand binding domain (262 to 507 aa) assessed as inhibition of SRC1-4 co-activator peptide recruit...More data for this Ligand-Target Pair
TargetNuclear receptor ROR-beta(Homo sapiens (Human))TBA
LigandPNGBDBM50005410(CHEMBL139197 | CHEMBL2137199)
Affinity DataIC50: >2.00E+4nMAssay Description:Inverse agonist activity at human GAL4-fused RORbeta LBD transfected in 293T cell measured after 24 hrs by dual luciferase assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50005410(CHEMBL139197 | CHEMBL2137199)
Affinity DataIC50: >2.00E+4nMAssay Description:Inverse agonist activity at human GAL4-fused LXRalpha LBD transfected in 293T cell measured after 24 hrs by dual luciferase assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBile acid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50005410(CHEMBL139197 | CHEMBL2137199)
Affinity DataIC50: >2.00E+4nMAssay Description:Inverse agonist activity at human GAL4-fused FXR LBD transfected in 293T cell measured after 24 hrs by dual luciferase assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNuclear receptor ROR-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50005410(CHEMBL139197 | CHEMBL2137199)
Affinity DataIC50: >2.00E+4nMAssay Description:Inverse agonist activity at human GAL4-fused RORalpha LBD transfected in 293T cell measured after 24 hrs by dual luciferase assayMore data for this Ligand-Target Pair
In DepthDetails PubMed