Affinity DataIC50: 600nMAssay Description:Inhibitory activity against type IIA sodium channel in CNaIIA-1 cell line expressed in CHO cellsMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Chonnam National University
Curated by ChEMBL
Chonnam National University
Curated by ChEMBL
Affinity DataIC50: 1.07E+3nMAssay Description:Inhibition of yeast Farnesyl transferaseMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Chonnam National University
Curated by ChEMBL
Chonnam National University
Curated by ChEMBL
Affinity DataIC50: 1.07E+3nMAssay Description:Inhibition of [3H]dopamine uptake at DAT (unknown origin)More data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Chonnam National University
Curated by ChEMBL
Chonnam National University
Curated by ChEMBL
Affinity DataIC50: 2.21E+3nMAssay Description:Inhibition of [3H]norepinephrine uptake at NET (unknown origin)More data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Chonnam National University
Curated by ChEMBL
Chonnam National University
Curated by ChEMBL
Affinity DataIC50: 2.21E+3nMAssay Description:Inhibition of [3H]-5-norepinephrine reuptake in human NET expressed in HEK293 cells by microbeta liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Chonnam National University
Curated by ChEMBL
Chonnam National University
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of [3H]serotonin uptake at SERT (unknown origin)More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Chonnam National University
Curated by ChEMBL
Chonnam National University
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of [3H]-5-hydroxytryptamine reuptake in human SERT expressed in HEK293 cells by microbeta liquid scintillation counting methodMore data for this Ligand-Target Pair