TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
Reckitt & Colman
Curated by ChEMBL
Reckitt & Colman
Curated by ChEMBL
Affinity DataIC50: 78nMAssay Description:Inhibitory activity against Alpha-2 adrenergic receptor in rat vas deferensMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
Reckitt & Colman
Curated by ChEMBL
Reckitt & Colman
Curated by ChEMBL
Affinity DataIC50: 520nMAssay Description:50% inhibition of specific [3H]clonidine binding (0.4 nM) to Alpha-2 adrenergic receptors in rat isolated brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of specific [3H]prazosin binding (0.2 nM) to rat brain membranes alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: >1.19E+6nMAssay Description:Inhibition of HIV1 RTMore data for this Ligand-Target Pair