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Found 7 of ic50 for monomerid = 50100615
TargetEphrin type-A receptor 2 [596-900](Homo sapiens (Human))
Technical University of Munich

LigandPNGBDBM50100615(E-7050 | E7050 | Golvatinib)
Affinity DataIC50:  13nMAssay Description:Refer to Reaction Biology Corps.More data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50100615(E-7050 | E7050 | Golvatinib)
Affinity DataIC50:  14nMAssay Description:Inhibition of c-Met autophosphorylation in human MKN45 cells after 2 hrs by Western blot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50100615(E-7050 | E7050 | Golvatinib)
Affinity DataIC50:  14nMAssay Description:Inhibition of MET autophosphorylation in human MKN45 cells after 2 hrs by Western blot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
St. John'S University

Curated by ChEMBL
LigandPNGBDBM50100615(E-7050 | E7050 | Golvatinib)
Affinity DataIC50:  16nMAssay Description:Inhibition of VEGF induced VEGFR2 phosphorylation in HUVEC preincubated for 1 hr followed by VEGF-stimulation for 5 mins by Western blot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
St. John'S University

Curated by ChEMBL
LigandPNGBDBM50100615(E-7050 | E7050 | Golvatinib)
Affinity DataIC50:  16nMAssay Description:Inhibition of VEGFR-2 autophosphorylation in HUVEC after 1 hr by Western blot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50100615(E-7050 | E7050 | Golvatinib)
Affinity DataIC50:  20nMAssay Description:Inhibition of human recombinant c-Met pre-incubated for 5 mins before ATP/substrate peptide cocktail addition measured after 30 mins by colorimetric ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
St. John'S University

Curated by ChEMBL
LigandPNGBDBM50100615(E-7050 | E7050 | Golvatinib)
Affinity DataIC50:  40nMAssay Description:Inhibition of human recombinant VEGFR2 pre-incubated for 5 mins before ATP/substrate peptide cocktail addition measured after 30 mins by colorimetric...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed