Compile Data Set for Download or QSAR
maximum 50k data
Found 4 of ic50 for monomerid = 50115617
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50115617(CHEMBL3609257)
Affinity DataIC50:  0.207nMAssay Description:Antagonist activity at human Kv1.3 expressed in CHOK1 cells assessed as inhibition of potassium currents after 10 mins by IonWorks Quattro patch clam...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50115617(CHEMBL3609257)
Affinity DataIC50:  0.357nMAssay Description:Antagonist activity at Kv1.3 in human whole blood assessed as inhibition of thapsigargin-induced IL-2 secretion incubated for 30 prior to thapsigargi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50115617(CHEMBL3609257)
Affinity DataIC50:  0.573nMAssay Description:Antagonist activity at Kv1.3 in human whole blood assessed as inhibition of thapsigargin-induced IFN-gamma secretion incubated for 30 prior to thapsi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50115617(CHEMBL3609257)
Affinity DataIC50:  1.02nMAssay Description:Antagonist activity at human Kv1.1 expressed in HEK293 cells assessed as inhibition of potassium currents after 10 mins by IonWorks Quattro patch cla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed