Affinity DataIC50: 180nMAssay Description:Concentration required to inhibit the maximum [14C]-Gly-Sar uptake by human Intestinal peptide transporter PepT1 in Caco-2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:50% Inhibitory potency against enkephalinase from mouse striatum.More data for this Ligand-Target Pair
Affinity DataIC50: 7.00E+4nMAssay Description:Binding affinity to human PEPT1 assessed as inhibition of [14C]Gly-Sar uptake in MDCK cellsMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+6nMAssay Description:50% Inhibitory potency against Angiotensin I converting enzyme from mouse striatum.More data for this Ligand-Target Pair