Compile Data Set for Download or QSAR
maximum 50k data
Found 2 of ic50 for monomerid = 50146685
TargetEndothelin-1 receptor(Homo sapiens (Human))
Actelion Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50146685((S)-(4,6-Dimethyl-pyrimidin-2-yloxy)-[(S)-1-(4-met...)
Affinity DataIC50:  4.60nMAssay Description:Antagonist activity towards human recombinant Endothelin A receptor expressed in chinese hamster ovary (CHO) cells determined using [125I]-ET-1 as ra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50146685((S)-(4,6-Dimethyl-pyrimidin-2-yloxy)-[(S)-1-(4-met...)
Affinity DataIC50:  22.4nMAssay Description:Antagonist activity towards human recombinant Endothelin B receptor expressed in chinese hamster ovary (CHO) cells determined using [125I]-ET-1 as ra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed