TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Affinity DataIC50: 397nMAssay Description:Activity at human mGluR5 assessed as effect on glutamate-induced calcium ion mobilization by FLIPRMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Astrazeneca R & D M£Lndal
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Activity at human mGluR1 assessed as effect on glutamate-induced calcium ion mobilization by FLIPRMore data for this Ligand-Target Pair