TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
RhôNe-Poulenc Rorer
Curated by ChEMBL
RhôNe-Poulenc Rorer
Curated by ChEMBL
Affinity DataIC50: 0.130nMAssay Description:Inhibition of human recombinant PDE4B1 assessed as reduction in [3H]cAMP hydrolysis to [3H]AMP incubated for 60 mins by PDE-SPA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Antagonist activity at adenosine A1 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Antagonist activity at adenosine A2a receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 169nMAssay Description:Antagonist activity at adenosine A2b receptor (unknown origin)More data for this Ligand-Target Pair