Compile Data Set for Download or QSAR
maximum 50k data
Found 3 of ic50 for monomerid = 50249208
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
California Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50249208(2-methoxy-4-(2-nitrovinyl)phenyl benzoate | CHEMBL...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of His6-tagged p97 (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as reduction in ATPase activity measured after 60 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50249208(2-methoxy-4-(2-nitrovinyl)phenyl benzoate | CHEMBL...)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibition of recombinant Syk (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))
California Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50249208(2-methoxy-4-(2-nitrovinyl)phenyl benzoate | CHEMBL...)
Affinity DataIC50:  5.70E+3nMAssay Description:Inhibition of p97 in human HeLa cells assessed as reduction in proteasomal turnover of p97-dependent reporter substrate UbG76V-GFP incubated for 120 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed