Compile Data Set for Download or QSAR
maximum 50k data
Found 5 of ic50 for monomerid = 50268875
TargetP2X purinoceptor 2(RAT)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50268875(CHEMBL496401 | Sodium 1-amino-4-[4-(4,6-dichloro-[...)
Affinity DataIC50:  117nMAssay Description:Antagonist activity against rat P2X2 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 6(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50268875(CHEMBL496401 | Sodium 1-amino-4-[4-(4,6-dichloro-[...)
Affinity DataIC50:  1.00E+4nMAssay Description:Antagonist activity against human P2Y6 receptor expressed in 1321N1 astrocytoma cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50268875(CHEMBL496401 | Sodium 1-amino-4-[4-(4,6-dichloro-[...)
Affinity DataIC50:  1.00E+4nMAssay Description:Antagonist activity against human P2Y4 receptor expressed in 1321N1 astrocytoma cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(RAT)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50268875(CHEMBL496401 | Sodium 1-amino-4-[4-(4,6-dichloro-[...)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50268875(CHEMBL496401 | Sodium 1-amino-4-[4-(4,6-dichloro-[...)
Affinity DataIC50:  1.21E+4nMAssay Description:Antagonist activity against human P2Y2 receptor expressed in 1321N1 astrocytoma cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed