Compile Data Set for Download or QSAR
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Found 3 of ic50 for monomerid = 50273896
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50273896(CHEMBL453249 | tert-Butyl-4-[1-pyridin-3-yl-1 H-1,...)
Affinity DataIC50:  55nMAssay Description:Antagonist activity at human mGluR1 expressed in CHO cells assessed as calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Mus musculus)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50273896(CHEMBL453249 | tert-Butyl-4-[1-pyridin-3-yl-1 H-1,...)
Affinity DataIC50:  180nMAssay Description:Antagonist activity at mouse mGluR1 expressed in CHO cells assessed as calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50273896(CHEMBL453249 | tert-Butyl-4-[1-pyridin-3-yl-1 H-1,...)
Affinity DataIC50:  8.30E+3nMAssay Description:Antagonist activity at human mGluR5 expressed in CHO cells assessed as calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed