Compile Data Set for Download or QSAR
maximum 50k data
Found 3 of ic50 for monomerid = 50273897
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50273897(CHEMBL457873 | tert-Butyl-4-[1-pyridin-4-yl-1 H-1,...)
Affinity DataIC50:  220nMAssay Description:Antagonist activity at human mGluR1 expressed in CHO cells assessed as calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Mus musculus)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50273897(CHEMBL457873 | tert-Butyl-4-[1-pyridin-4-yl-1 H-1,...)
Affinity DataIC50:  1.00E+3nMAssay Description:Antagonist activity at mouse mGluR1 expressed in CHO cells assessed as calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50273897(CHEMBL457873 | tert-Butyl-4-[1-pyridin-4-yl-1 H-1,...)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at human mGluR5 expressed in CHO cells assessed as calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed