Compile Data Set for Download or QSAR
maximum 50k data
Found 2 of ic50 for monomerid = 50293873
TargetB2 bradykinin receptor(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50293873(5-(8-((3,5-dichloropyridin-4-yl)methoxy)-2-methylq...)
Affinity DataIC50:  135nMAssay Description:Displacement of [3H]bradykinin from human recombinant B2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50293873(5-(8-((3,5-dichloropyridin-4-yl)methoxy)-2-methylq...)
Affinity DataIC50:  420nMAssay Description:Antagonist activity at B2 receptor in human HF15 cells assessed as inhibition of bradykinin-induced calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed