Compile Data Set for Download or QSAR
maximum 50k data
Found 7 of ic50 for monomerid = 50336767
TargetP2X purinoceptor 2(RAT)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50336767(CHEMBL257495 | PSB-716 | sodium 1-amino-4-(2-metho...)
Affinity DataIC50:  2.00E+3nMAssay Description:Antagonist activity against rat P2X2 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50336767(CHEMBL257495 | PSB-716 | sodium 1-amino-4-(2-metho...)
Affinity DataIC50:  3.98E+3nMAssay Description:Antagonist activity at human P2Y4 receptor transfected in human 1321N1 cells assessed as inhibition of UTP-activated intracellular calcium mobilizati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Mus musculus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50336767(CHEMBL257495 | PSB-716 | sodium 1-amino-4-(2-metho...)
Affinity DataIC50:  9.00E+3nMAssay Description:Antagonist activity at mouse P2Y2 receptor in mouse NG108-15 cells assessed as inhibition of UTP-induced calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50336767(CHEMBL257495 | PSB-716 | sodium 1-amino-4-(2-metho...)
Affinity DataIC50:  9.82E+3nMAssay Description:Antagonist activity at human recombinant P2Y2 receptor in 1321N1 cells assessed as inhibition of UTP-induced calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(RAT)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50336767(CHEMBL257495 | PSB-716 | sodium 1-amino-4-(2-metho...)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50336767(CHEMBL257495 | PSB-716 | sodium 1-amino-4-(2-metho...)
Affinity DataIC50:  5.00E+4nMAssay Description:Antagonist activity at human P2Y4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 6(Rattus norvegicus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50336767(CHEMBL257495 | PSB-716 | sodium 1-amino-4-(2-metho...)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at rat P2Y6 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed