Compile Data Set for Download or QSAR
maximum 50k data
Found 2 of ic50 for monomerid = 50340441
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Sanofi-Aventis R&D

Curated by ChEMBL
LigandPNGBDBM50340441((3-(1H-pyrazol-4-yl)pyrrolidin-1-yl)(2H-benzo[b][1...)
Affinity DataIC50:  27nMAssay Description:Inhibition of human recombinant 11beta-HSD1 assessed as conversion of radiolabelled-cortisone to cortisol by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Sanofi-Aventis R&D

Curated by ChEMBL
LigandPNGBDBM50340441((3-(1H-pyrazol-4-yl)pyrrolidin-1-yl)(2H-benzo[b][1...)
Affinity DataIC50:  490nMAssay Description:Inhibition of mouse recombinant 11beta-HSD1 assessed as conversion of radiolabelled-cortisone to cortisol by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed