Compile Data Set for Download or QSAR
maximum 50k data
Found 4 of ic50 for monomerid = 50583764
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Servier Research Institute Of Medicinal Chemistry

Curated by ChEMBL
LigandPNGBDBM50583764(CHEMBL5084166)
Affinity DataIC50:  5nMAssay Description:Inhibition of DYRK1A (unknown origin) using Ulight-MBP as substrate and ATP as co-substrate incubated for 40 mins and measured after 1 hr by TR-FRET ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Servier Research Institute Of Medicinal Chemistry

Curated by ChEMBL
LigandPNGBDBM50583764(CHEMBL5084166)
Affinity DataIC50:  44nMAssay Description:Inhibition of wild type full length DYRK1A (unknown origin) in human U2OS cells assessed as reduction in pSER520 autophosphorylation incubated for 5 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 2(Homo sapiens (Human))
Servier Research Institute Of Medicinal Chemistry

Curated by ChEMBL
LigandPNGBDBM50583764(CHEMBL5084166)
Affinity DataIC50:  195nMAssay Description:Inhibition of DYRK2 (unknown origin) using Ulight-MBP as substrate and ATP as co-substrate incubated for 40 mins and measured after 1 hr by TR-FRET a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Servier Research Institute Of Medicinal Chemistry

Curated by ChEMBL
LigandPNGBDBM50583764(CHEMBL5084166)
Affinity DataIC50:  467nMAssay Description:Inhibition of CDK9 (unknown origin) using Ulight-MBP as substrate and ATP as co-substrate incubated for 40 mins and measured after 1 hr by TR-FRET as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed