Compile Data Set for Download or QSAR
maximum 50k data
Found 3 of ic50 for monomerid = 7338
TargetGlycogen synthase kinase-3 beta(Rattus norvegicus (rat))
Universitat Hamburg

LigandPNGBDBM7338(13-chloro-3-thia-7,17-diazatetracyclo[8.7.0.0^{2,6...)
Affinity DataIC50:  400nMT: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/ [gamma-32P] ATP. 32...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 1/G2/mitotic-specific cyclin-B(Marthasterias glacialis (starfish))
Universitat Hamburg

LigandPNGBDBM7338(13-chloro-3-thia-7,17-diazatetracyclo[8.7.0.0^{2,6...)
Affinity DataIC50:  500nMT: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/ [gamma-32P] ATP. 32...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1 [99-307](Homo sapiens (Human))
Universitat Hamburg

LigandPNGBDBM7338(13-chloro-3-thia-7,17-diazatetracyclo[8.7.0.0^{2,6...)
Affinity DataIC50:  5.00E+3nMT: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/ [gamma-32P] ATP. 32...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed