Compile Data Set for Download or QSAR
maximum 50k data
Found 4 of ic50 for monomerid = 7515
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Institut Curie

Curated by ChEMBL
LigandPNGBDBM7515(2,6,9-Trisubstituted purine deriv. 10 | [(2R)-1-[6...)
Affinity DataIC50:  650nMAssay Description:Inhibition of cyclin-dependent kinase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 1/G2/mitotic-specific cyclin-B(Marthasterias glacialis (starfish))
Institut Curie

LigandPNGBDBM7515(2,6,9-Trisubstituted purine deriv. 10 | [(2R)-1-[6...)
Affinity DataIC50:  650nMT: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/ [gamma-32P] ATP. 32...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
Institut Curie

Curated by ChEMBL
LigandPNGBDBM7515(2,6,9-Trisubstituted purine deriv. 10 | [(2R)-1-[6...)
Affinity DataIC50:  1.30E+3nMAssay Description:Compound was tested for its inhibitory activity against cyclin-dependent kinase 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Institut Curie

LigandPNGBDBM7515(2,6,9-Trisubstituted purine deriv. 10 | [(2R)-1-[6...)
Affinity DataIC50:  1.30E+3nMT: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/ [gamma-32P] ATP. 32...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed