Affinity DataKd: 620nMAssay Description:Binding affinity to human C-terminal His8-tagged JAK2 pseudokinase (513 to 827 residues) expressed in baculovirus infected Hi-5 cells by intrinsic tr...More data for this Ligand-Target Pair
Affinity DataKd: 2.00E+3nMAssay Description:Binding affinity to wild type human C-terminal thrombin cleavage site-fused/ 6xHis-tagged JAK2 JH2 pseudokinase domain (536 to 812 residues) expresse...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
Affinity DataKd: 3.50E+3nMAssay Description:Binding affinity to BRD4 bromodomain 1 (unknown origin) by ITC assayMore data for this Ligand-Target Pair
Affinity DataKd: 3.55E+3nMAssay Description:Binding affinity to human RSK1 assessed as dissociation constantMore data for this Ligand-Target Pair