Affinity DataKd: 0.550nMAssay Description:Binding constant for ALK kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.10nMAssay Description:Binding constant for LTK kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.70nMAssay Description:Binding constant for INSR kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 7nMAssay Description:Binding constant for IGF1R kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 8.60nMAssay Description:Binding constant for INSRR kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 9.30nMAssay Description:Binding constant for FER kinase domainMore data for this Ligand-Target Pair
TargetMyosin light chain kinase, smooth muscle(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 11nMAssay Description:Binding constant for MYLK kinase domainMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase ROS(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 15nMAssay Description:Binding constant for ROS1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 16nMAssay Description:Binding constant for CLK2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 21nMAssay Description:Binding constant for CLK1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 47nMAssay Description:Binding constant for PLK1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 52nMAssay Description:Binding constant for FES kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 60nMAssay Description:Binding constant for CLK4 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 70nMAssay Description:Binding constant for STK33 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 74nMAssay Description:Binding constant for EGFR(T790M) kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 76nMAssay Description:Binding constant for TTK kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 76nMAssay Description:Binding constant for PYK2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 130nMAssay Description:Binding constant for JNK3 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 150nMAssay Description:Binding constant for EGFR(L858R,T790M) kinase domainMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 170nMAssay Description:Binding constant for LRRK2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 170nMAssay Description:Binding constant for RSK2(Kin.Dom.1-N-terminal) kinase domainMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 19(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 190nMAssay Description:Binding constant for YSK4 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 200nMAssay Description:Binding constant for FAK kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 210nMAssay Description:Binding constant for JNK1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 270nMAssay Description:Binding constant for GAK kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 280nMAssay Description:Binding constant for CHEK2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 300nMAssay Description:Binding constant for AXL kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 410nMAssay Description:Binding constant for PRKD3 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 410nMAssay Description:Binding constant for RSK1(Kin.Dom.1-N-terminal) kinase domainMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type IV(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 470nMAssay Description:Binding constant for CAMK4 kinase domainMore data for this Ligand-Target Pair
TargetTestis-specific serine/threonine-protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 470nMAssay Description:Binding constant for TSSK1B kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 520nMAssay Description:Binding constant for JNK2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 540nMAssay Description:Binding constant for GRK7 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 620nMAssay Description:Binding constant for DAPK1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 650nMAssay Description:Binding constant for PRKD1 kinase domainMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 730nMAssay Description:Binding constant for LRRK2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 780nMAssay Description:Binding constant for CSNK1E kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 830nMAssay Description:Binding constant for GRK1 kinase domainMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 910nMAssay Description:Binding constant for MEK4 kinase domainMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 970nMAssay Description:Binding constant for DYRK1B kinase domainMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 3(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 1.00E+3nMAssay Description:Binding constant for MEK3 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.10E+3nMAssay Description:Binding constant for DAPK2 kinase domainMore data for this Ligand-Target Pair
TargetPhosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 1.10E+3nMAssay Description:Binding constant for PHKG1 kinase domainMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 1.20E+3nMAssay Description:Binding constant for DYRK1A kinase domainMore data for this Ligand-Target Pair
TargetHomeodomain-interacting protein kinase 4(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 1.20E+3nMAssay Description:Binding constant for HIPK4 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.20E+3nMAssay Description:Binding constant for DAPK3 kinase domainMore data for this Ligand-Target Pair
TargetHomeodomain-interacting protein kinase 2(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 1.20E+3nMAssay Description:Binding constant for HIPK2 kinase domainMore data for this Ligand-Target Pair
TargetHomeodomain-interacting protein kinase 1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 1.30E+3nMAssay Description:Binding constant for HIPK1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.40E+3nMAssay Description:Binding constant for EGFR(L861Q) kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.40E+3nMAssay Description:Binding constant for TAOK3 kinase domainMore data for this Ligand-Target Pair