TargetProto-oncogene tyrosine-protein kinase ROS(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 0.490nMAssay Description:Binding constant for ROS1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 0.830nMAssay Description:Binding constant for ULK1 kinase domainMore data for this Ligand-Target Pair
TargetBone morphogenetic protein receptor type-1B(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 0.850nMAssay Description:Binding constant for BMPR1B kinase domainMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 0.860nMAssay Description:Binding constant for LRRK2(G2019S) kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 0.930nMAssay Description:Binding constant for PLK4 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 0.950nMAssay Description:Binding constant for LTK kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.10nMAssay Description:Binding constant for ALK kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.10nMAssay Description:Binding constant for FAK kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.10nMAssay Description:Binding constant for PYK2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.20nMAssay Description:Binding constant for SNARK kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.20nMAssay Description:Binding affinity to NUAK2 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 1.40nMAssay Description:Binding constant for LRRK2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.40nMAssay Description:Binding constant for FER kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.80nMAssay Description:Binding constant for ULK2 kinase domainMore data for this Ligand-Target Pair
TargetNon-receptor tyrosine-protein kinase TNK1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 1.80nMAssay Description:Binding constant for TNK1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 2nMAssay Description:Binding constant for TNK2 kinase domainMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 2nMAssay Description:Binding constant for FLT3(D835Y) kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 2.40nMAssay Description:Binding constant for INSR kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 2.70nMAssay Description:Binding constant for IGF1R kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 3.20nMAssay Description:Binding constant for STK33 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 3.40nMAssay Description:Binding constant for EGFR(L858R,T790M) kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 4.80nMAssay Description:Binding constant for FES kinase domainMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 4.90nMAssay Description:Binding constant for FLT3(D835H) kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 4.90nMAssay Description:Binding constant for DCAMKL1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 5.30nMAssay Description:Binding constant for GAK kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 5.40nMAssay Description:Binding constant for ABL1(T315I)-phosphorylated kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 6.20nMAssay Description:Binding constant for INSRR kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 7.10nMAssay Description:Binding constant for EGFR(T790M) kinase domainMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 8.20nMAssay Description:Binding constant for FLT3(D835Y) kinase domainMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 8.60nMAssay Description:Binding constant for FLT3(ITD) kinase domainMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 11nMAssay Description:Binding constant for FLT3(N841I) kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 11nMAssay Description:Binding constant for ULK3 kinase domainMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase kinase 2(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 11nMAssay Description:Binding constant for CAMKK2 kinase domainMore data for this Ligand-Target Pair
TargetMAP/microtubule affinity-regulating kinase 4(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 12nMAssay Description:Binding constant for MARK4 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 12nMAssay Description:Inhibition AXL (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 12nMAssay Description:Binding constant for CLK1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 12nMAssay Description:Binding constant for AXL kinase domainMore data for this Ligand-Target Pair
TargetMAP/microtubule affinity-regulating kinase 3(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 12nMAssay Description:Binding constant for MARK3 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 13nMAssay Description:Binding constant for ARK5 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 13nMAssay Description:Binding constant for YANK1 kinase domainMore data for this Ligand-Target Pair
TargetPhosphorylase b kinase gamma catalytic chain, liver/testis isoform(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 13nMAssay Description:Binding constant for PHKG2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 13nMAssay Description:Binding affinity to NUAK1 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 14nMAssay Description:Binding constant for ABL1(F317I)-phosphorylated kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 14nMAssay Description:Binding constant for DCAMKL3 kinase domainMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor Tie-1(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 15nMAssay Description:Binding constant for TIE1 kinase domainMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 15nMAssay Description:Binding constant for FLT3 kinase domainMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Ambit Biosciences
Curated by ChEMBL
Ambit Biosciences
Curated by ChEMBL
Affinity DataKd: 15nMAssay Description:Binding affinity to human FLT3More data for this Ligand-Target Pair
Affinity DataKd: 15nMAssay Description:Binding constant for SIK kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 16nMAssay Description:Binding constant for JAK2(JH1domain-catalytic) kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 16nMAssay Description:Binding constant for DCAMKL2 kinase domainMore data for this Ligand-Target Pair