Affinity DataKd: 90nMAssay Description:Binding affinity to AhR (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 90nMAssay Description:Displacement of 2-azido-3-[125I]7,8-dibromodibenzo-pdioxin from C57BL/6J mouse liver AhRMore data for this Ligand-Target Pair
TargetDNA topoisomerase type IB small subunit(Leishmania donovani)
India Institute Of Chemical Biology
Curated by ChEMBL
India Institute Of Chemical Biology
Curated by ChEMBL
Affinity DataKd: 3.80E+5nMAssay Description:Binding affinity to recombinant drug-resistant Leishmania donovani LdDR50 topoisomerase 1b small subunit N184S mutant after 24 hrs by equilibrium dia...More data for this Ligand-Target Pair
Affinity DataKd: 5.30E+5nMAssay Description:Binding affinity to recombinant drug-resistant Leishmania donovani LdDR50 topoisomerase 1b large subunit F270L mutant after 24 hrs by equilibrium dia...More data for this Ligand-Target Pair
Affinity DataKd: 7.60E+5nMAssay Description:Binding affinity to recombinant drug-resistant Leishmania donovani LdDR50 topoisomerase 1b large subunit F270L, K430N mutant after 24 hrs by equilibr...More data for this Ligand-Target Pair