Compile Data Set for Download or QSAR
maximum 50k data
Found 2 of ki for monomerid = 1201
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Sandoz Forschungsinstitut Ges.M.B.H.

Curated by ChEMBL
LigandPNGBDBM1201(2-Aminobenzyl-Substituted AHPPA deriv. 18 | tert-b...)
Affinity DataKi:  79.4nMAssay Description:Inhibitory activity was determined against HIV type 1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Sandoz Research Institute

LigandPNGBDBM1201(2-Aminobenzyl-Substituted AHPPA deriv. 18 | tert-b...)
Affinity DataKi:  80nM ΔG°:  -42.1kJ/mole IC50:  4.00E+3nMpH: 6.25 T: 2°CAssay Description:Enzymatic activity was measured by following cleavage of the substrate H-Lys-Ala-Arg-Val-Leu-pNph-Glu-Ala-Nle-NH2. Products of the cleavage reaction ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed