Compile Data Set for Download or QSAR
maximum 50k data
Found 4 of ki for monomerid = 175380
TargetAdenosine receptor A2a(Homo sapiens (Human))
Panjab University

LigandPNGBDBM175380(1,3-Dimethyl-8-[3-{2-(piperidin-1-yl)]-2-oxoethoxy...)
Affinity DataKi:  209nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Panjab University

LigandPNGBDBM175380(1,3-Dimethyl-8-[3-{2-(piperidin-1-yl)]-2-oxoethoxy...)
Affinity DataKi:  1.52E+3nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Panjab University

LigandPNGBDBM175380(1,3-Dimethyl-8-[3-{2-(piperidin-1-yl)]-2-oxoethoxy...)
Affinity DataKi:  4.04E+3nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3 [I248L](Homo sapiens (Human))
Panjab University

LigandPNGBDBM175380(1,3-Dimethyl-8-[3-{2-(piperidin-1-yl)]-2-oxoethoxy...)
Affinity DataKi:  4.16E+3nMAssay Description:Dissociation constants at A1, A2A and A3 receptors (Ki-values) were determined in radioligand competition experiments as reported earlier [19,20]. Al...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed