Compile Data Set for Download or QSAR
maximum 50k data
Found 6 of ki for monomerid = 50000407
TargetBeta-lactamase(Aeromonas hydrophila)
Universit£

Curated by ChEMBL
LigandPNGBDBM50000407(2-carboxypyridine | CHEMBL72628 | alpha-picolinic ...)
Affinity DataKi:  5.70E+3nMAssay Description:Inhibition of Aeromonas hydrophila beta lactamase CphA by competitive inhibition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Aeromonas hydrophila)
Universit£

Curated by ChEMBL
LigandPNGBDBM50000407(2-carboxypyridine | CHEMBL72628 | alpha-picolinic ...)
Affinity DataKi:  4.60E+4nMAssay Description:Inhibition of Aeromonas hydrophila beta lactamase CphA at pH 7.0More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Aeromonas hydrophila)
Universit£

Curated by ChEMBL
LigandPNGBDBM50000407(2-carboxypyridine | CHEMBL72628 | alpha-picolinic ...)
Affinity DataKi:  7.60E+4nMAssay Description:Inhibition of Aeromonas hydrophila beta lactamase CphA at pH 8.0More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Aeromonas hydrophila)
Universit£

Curated by ChEMBL
LigandPNGBDBM50000407(2-carboxypyridine | CHEMBL72628 | alpha-picolinic ...)
Affinity DataKi:  4.40E+5nMAssay Description:Inhibition of Aeromonas hydrophila beta lactamase CphA at pH 9.0More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Aeromonas hydrophila)
Universit£

Curated by ChEMBL
LigandPNGBDBM50000407(2-carboxypyridine | CHEMBL72628 | alpha-picolinic ...)
Affinity DataKi:  1.10E+6nMAssay Description:Inhibition of Aeromonas hydrophila beta lactamase CphA at pH 10.0More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProton-coupled amino acid transporter 1(Homo sapiens (Human))
Martin-Luther-University Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50000407(2-carboxypyridine | CHEMBL72628 | alpha-picolinic ...)
Affinity DataKi:  1.80E+7nMAssay Description:Inhibition of human PAT1-mediated L-[3H]proline uptake in human Caco2 cells after 10 mins by liquid scintillation countingChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed