Compile Data Set for Download or QSAR
maximum 50k data
Found 3 of ki for monomerid = 50089084
TargetCarbapenem-hydrolyzing beta-lactamase KPC()
Qpex Biopharma

Curated by ChEMBL
LigandPNGBDBM50089084(CHEMBL3317857 | Vaborbactam)
Affinity DataKi:  56nMAssay Description:Inhibition of recombinant Escherichia coli KPC-2 using nitrocefin as substrate preincubated for 10 mins followed by substrate addition and measured e...More data for this Ligand-Target Pair
TargetOXA23 carbapenemase(Acinetobacter baumannii)
Qpex Biopharma

Curated by ChEMBL
LigandPNGBDBM50089084(CHEMBL3317857 | Vaborbactam)
Affinity DataKi: >4.00E+4nMAssay Description:Inhibition of Acinetobacter baumannii OXA-23 using nitrocefin as substrate preincubated for 10 mins followed by substrate addition measured every 10 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVIM-1 metallo-beta-lactamase(Klebsiella pneumoniae)
Qpex Biopharma

Curated by ChEMBL
LigandPNGBDBM50089084(CHEMBL3317857 | Vaborbactam)
Affinity DataKi: >4.00E+4nMAssay Description:Inhibition of recombinant Escherichia coli VIM-1 using nitrocefin as substrate preincubated for 10 mins followed by substrate addition measured every...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed