Compile Data Set for Download or QSAR
maximum 50k data
Found 3 of ki for monomerid = 50090073
TargetBifunctional dihydrofolate reductase-thymidylate synthase(Plasmodium falciparum (isolate K1 / Thailand))
Università

Curated by ChEMBL
LigandPNGBDBM50090073(1-(4-Fluoro-phenyl)-1,6-dihydro-[1,3,5]triazine-2,...)
Affinity DataKi:  88nMAssay Description:Inhibition constant against Plasmodium falciparum dihydrofolate reductaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional dihydrofolate reductase-thymidylate synthase(Plasmodium falciparum)
National Center For Genetic Engineering And Biotechnology At Thailand

Curated by ChEMBL
LigandPNGBDBM50090073(1-(4-Fluoro-phenyl)-1,6-dihydro-[1,3,5]triazine-2,...)
Affinity DataKi:  270nMAssay Description:Evaluated for inhibition constant (Ki wt) against Wild-type dihydrofolate reductase of Plasmodium falciparumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional dihydrofolate reductase-thymidylate synthase [A16V,S108T](Plasmodium falciparum)
National Center For Genetic Engineering And Biotechnology At Thailand

Curated by ChEMBL
LigandPNGBDBM50090073(1-(4-Fluoro-phenyl)-1,6-dihydro-[1,3,5]triazine-2,...)
Affinity DataKi:  469nMAssay Description:Inhibition constant (Ki mut) against A16V+S108T Mutant DHFRs of Plasmodium falciparumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed