Affinity DataKi: 0.150nMAssay Description:Binding affinity against adenosine A1 receptor in bovine cortical membranes using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.150nMAssay Description:Ability to displace the specific binding of [3H]CHA to adenosine A1 receptor from bovine brain cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.62nMAssay Description:Displacement of [3H]-DPCPX from adenosine A1 receptor in bovine brain cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Ability to displace the specific binding of [3H]-CGS- to adenosine A2A receptor form bovine brain striatal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Binding affinity against adenosine A2 receptor in bovine striatal membranes using [3H]-CGS-21,680 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Binding affinity against adenosine A1 receptor in human cortical membranes using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 450nMAssay Description:Binding affinity against adenosine A2 receptor in human striatal membranes using [3H]-CGS-21,680 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 670nMAssay Description:Displacement of [3H]-DPCPX from adenosine A1 receptor in human brain cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.10E+3nMAssay Description:Ability to displace the specific binding of [3H](R)-PIA to adenosine A3 receptor from rat testis membranesMore data for this Ligand-Target Pair