Compile Data Set for Download or QSAR
maximum 50k data
Found 8 of ki for monomerid = 50094695
TargetAdenosine receptor A3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50094695(1-(2-(furan-2-yl)-8-(3-methylbut-2-enyl)-8H-pyrazo...)
Affinity DataKi:  40nMAssay Description:Binding affinity for human adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50094695(1-(2-(furan-2-yl)-8-(3-methylbut-2-enyl)-8H-pyrazo...)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]-MRE3008-F20 from human adenosine A3 receptor expressed in CHO cells; range 35-47More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50094695(1-(2-(furan-2-yl)-8-(3-methylbut-2-enyl)-8H-pyrazo...)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50094695(1-(2-(furan-2-yl)-8-(3-methylbut-2-enyl)-8H-pyrazo...)
Affinity DataKi:  58nMAssay Description:Displacement of [3H]-DPCPX from Adenosine A2b receptor expressed in CHO cells; range 52-65More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50094695(1-(2-(furan-2-yl)-8-(3-methylbut-2-enyl)-8H-pyrazo...)
Affinity DataKi:  300nMAssay Description:Displacement of [3H]-DPCPX from human adenosine A1 receptor expressed in CHO cells; range 254-356More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50094695(1-(2-(furan-2-yl)-8-(3-methylbut-2-enyl)-8H-pyrazo...)
Affinity DataKi:  1.03E+3nMAssay Description:Displacement of [3H]-SCH- 58261 from human adenosine A2A receptor expressed in CHO cells; range 850-1230More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50094695(1-(2-(furan-2-yl)-8-(3-methylbut-2-enyl)-8H-pyrazo...)
Affinity DataKi:  1.03E+3nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50094695(1-(2-(furan-2-yl)-8-(3-methylbut-2-enyl)-8H-pyrazo...)
Affinity DataKi:  3.98E+4nMAssay Description:Displacement of [3H]MRE3008-F20 from human adenosine A3 receptor expressed in CHO cells after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed