TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-3/gamma-2(Homo sapiens (Human))
The Neuroscience Research Centre
Curated by ChEMBL
The Neuroscience Research Centre
Curated by ChEMBL
Affinity DataKi: 0.5nMAssay Description:Binding affinity at human recombinant gamma-aminobutyric-acid A receptor alpha3-beta3-gamma2 expressed in L(tk) cells by [3H]-Ro-15-1788 displacement...More data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Positive allosteric modulation of GABAA alpha3 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Positive allosteric modulation of GABAA alpha2 (unknown origin)More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Homo sapiens (Human))
The Neuroscience Research Centre
Curated by ChEMBL
The Neuroscience Research Centre
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Binding affinity at human recombinant gamma-aminobutyric-acid A receptor alpha1-beta3-gamma2 expressed in L(tk) cells by [3H]-Ro-15-1788 displacement...More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Positive allosteric modulation of GABAA alpha1 (unknown origin)More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-4(Homo sapiens (Human))
The Neuroscience Research Centre
Curated by ChEMBL
The Neuroscience Research Centre
Curated by ChEMBL
Affinity DataKi: 28nMAssay Description:Displacement of [3H]-Ro-15-1788 from human GABA-A receptor alpha4 subunit expressed in L(tk) cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-5(Homo sapiens (Human))
The Neuroscience Research Centre
Curated by ChEMBL
The Neuroscience Research Centre
Curated by ChEMBL
Affinity DataKi: 33nMAssay Description:Displacement of [3H]-Ro-15-1788 from human GABA-A receptor alpha5 subunit expressed in L(tk) cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-6(Homo sapiens (Human))
The Neuroscience Research Centre
Curated by ChEMBL
The Neuroscience Research Centre
Curated by ChEMBL
Affinity DataKi: 66nMAssay Description:Displacement of [3H]-Ro-15-1788 from human GABA-A receptor alpha6 subunit expressed in L(tk) cellsMore data for this Ligand-Target Pair