Compile Data Set for Download or QSAR
maximum 50k data
Found 4 of ki for monomerid = 50196139
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Timisoara Of The Romanian Academy

Curated by ChEMBL
LigandPNGBDBM50196139((3-methylquinolin-4-yl)-[4-(3,3,4-trimethylpiperaz...)
Affinity DataKi:  5.40nMAssay Description:Binding affinity to human cloned Alpha-2C adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Timisoara Of The Romanian Academy

Curated by ChEMBL
LigandPNGBDBM50196139((3-methylquinolin-4-yl)-[4-(3,3,4-trimethylpiperaz...)
Affinity DataKi:  5.40nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2C expressed in S115 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196139((3-methylquinolin-4-yl)-[4-(3,3,4-trimethylpiperaz...)
Affinity DataKi:  895nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2A expressed in S115 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Juvantia Pharma

Curated by ChEMBL
LigandPNGBDBM50196139((3-methylquinolin-4-yl)-[4-(3,3,4-trimethylpiperaz...)
Affinity DataKi:  1.27E+3nMAssay Description:Displacement of [3H]rauwolscine from human ADRA2B expressed in S115 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed