Compile Data Set for Download or QSAR
maximum 50k data
Found 4 of ki for monomerid = 50399568
TargetAdenosine receptor A3(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50399568(CHEMBL2180935)
Affinity DataKi:  1.99nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50399568(CHEMBL2180935)
Affinity DataKi:  75.4nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50399568(CHEMBL2180935)
Affinity DataKi:  322nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50399568(CHEMBL2180935)
Affinity DataKi:  2.62E+3nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as NECA-induced adenylate cyclase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed