Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with Target = 'Bombesin receptor subtype-3' and Ligand = 'BDBM50381914'
TargetBombesin receptor subtype-3(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50381914(MK-7725 | CHEMBL2023109)
Affinity DataEC50:  73nMAssay Description:Agonist activity at human BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Mouse)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50381914(MK-7725 | CHEMBL2023109)
Affinity DataEC50:  130nMAssay Description:Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Mouse)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50381914(MK-7725 | CHEMBL2023109)
Affinity DataEC50:  130nMAssay Description:Agonist activity at mouse BRS-3 expressed in HEK293AEQ cells assessed as bioluminescence for 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Mouse)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50381914(MK-7725 | CHEMBL2023109)
Affinity DataEC50:  22nMAssay Description:Agonist activity at mouse BRS-3 expressed in CHOK1 cells after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50381914(MK-7725 | CHEMBL2023109)
Affinity DataEC50:  1.40nMAssay Description:Agonist activity at human BRS-3 expressed in CHOK1 cells after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Mouse)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50381914(MK-7725 | CHEMBL2023109)
Affinity DataEC50:  130nMAssay Description:Agonist activity at mouse BRS3 expressed in human HEK293AEQ cells measured for 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50381914(MK-7725 | CHEMBL2023109)
Affinity DataEC50:  73nMAssay Description:Agonist activity at human BRS3 expressed in human HEK293AEQ cells measured for 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50381914(MK-7725 | CHEMBL2023109)
Affinity DataIC50: 3.60nMAssay Description:Displacement of [125I]-dY-peptide from human BRS-3 expressed in NFAT-CHO cells after 2 hrs by by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50381914(MK-7725 | CHEMBL2023109)
Affinity DataIC50: 3.60nMAssay Description:Displacement of 125I-dY-peptide from human BRS3 expressed in NFAT-CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed