Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with Target = 'D(2) dopamine receptor' and Ligand = 'BDBM81993'
TargetD(2) dopamine receptor(Human)
Neuroscience Research Centre

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 81993BDBM81993(Bromocriptine+ (GTP+) | BROMOCRIPTINE | Bromocript...)
Affinity DataKi:  0.620nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2012
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetD(2) dopamine receptor(Human)
Neuroscience Research Centre

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 81993BDBM81993(Bromocriptine+ (GTP+) | BROMOCRIPTINE | Bromocript...)
Affinity DataKi:  0.620nMAssay Description:Binding affinity to dopamine D2 receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetD(2) dopamine receptor(Mouse)
Medical Research Service

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 81993BDBM81993(Bromocriptine+ (GTP+) | BROMOCRIPTINE | Bromocript...)
Affinity DataKi:  0.690nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2011
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetD(2) dopamine receptor(Rat)
University of Pennsylvania

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 81993BDBM81993(Bromocriptine+ (GTP+) | BROMOCRIPTINE | Bromocript...)
Affinity DataKi:  0.800nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2011
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetD(2) dopamine receptor(Rat)
University of Pennsylvania

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 81993BDBM81993(Bromocriptine+ (GTP+) | BROMOCRIPTINE | Bromocript...)
Affinity DataKi:  0.800nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2011
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetD(2) dopamine receptor(Human)
Neuroscience Research Centre

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 81993BDBM81993(Bromocriptine+ (GTP+) | BROMOCRIPTINE | Bromocript...)
In Depth
Date in BDB:
3/3/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetD(2) dopamine receptor(Bovine)
TBA

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 81993BDBM81993(Bromocriptine+ (GTP+) | BROMOCRIPTINE | Bromocript...)
Affinity DataKi:  2.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2011
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetD(2) dopamine receptor(Rat)
University of Pennsylvania

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 81993BDBM81993(Bromocriptine+ (GTP+) | BROMOCRIPTINE | Bromocript...)
Affinity DataKd:  4nMAssay Description:In vitro affinity at mutant D2 receptor (S197A) in C6 (glioma) cell membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetD(2) dopamine receptor(Human)
Neuroscience Research Centre

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 81993BDBM81993(Bromocriptine+ (GTP+) | BROMOCRIPTINE | Bromocript...)
Affinity DataKi:  5.01nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetD(2) dopamine receptor(Rat)
University of Pennsylvania

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 81993BDBM81993(Bromocriptine+ (GTP+) | BROMOCRIPTINE | Bromocript...)
Affinity DataKi:  5.30nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2011
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetD(2) dopamine receptor(Rat)
University of Pennsylvania

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 81993BDBM81993(Bromocriptine+ (GTP+) | BROMOCRIPTINE | Bromocript...)
Affinity DataKi:  5.30nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2011
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetD(2) dopamine receptor(Rat)
University of Pennsylvania

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 81993BDBM81993(Bromocriptine+ (GTP+) | BROMOCRIPTINE | Bromocript...)
Affinity DataKd:  8nMAssay Description:In vitro affinity at wild type Dopamine receptor D2 on C6 (glioma) cell membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetD(2) dopamine receptor(Rat)
University of Pennsylvania

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 81993BDBM81993(Bromocriptine+ (GTP+) | BROMOCRIPTINE | Bromocript...)
Affinity DataKd:  8nMAssay Description:In vitro affinity at mutant D2 receptor (S194A) in C6 (glioma) cell membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetD(2) dopamine receptor(Human)
Neuroscience Research Centre

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 81993BDBM81993(Bromocriptine+ (GTP+) | BROMOCRIPTINE | Bromocript...)
Affinity DataKi:  8.20nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2012
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetD(2) dopamine receptor(Human)
Neuroscience Research Centre

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 81993BDBM81993(Bromocriptine+ (GTP+) | BROMOCRIPTINE | Bromocript...)
Affinity DataKi:  10nMAssay Description:Binding affinity towards Dopamine receptor D2 by displacement of [3H]U-86170.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetD(2) dopamine receptor(Human)
Neuroscience Research Centre

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 81993BDBM81993(Bromocriptine+ (GTP+) | BROMOCRIPTINE | Bromocript...)
Affinity DataKi:  12.6nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2011
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetD(2) dopamine receptor(Human)
Neuroscience Research Centre

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 81993BDBM81993(Bromocriptine+ (GTP+) | BROMOCRIPTINE | Bromocript...)
Affinity DataKi:  14.8nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetD(2) dopamine receptor(Human)
Neuroscience Research Centre

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 81993BDBM81993(Bromocriptine+ (GTP+) | BROMOCRIPTINE | Bromocript...)
Affinity DataKi:  15nMAssay Description:Displacement of [125]iodosulpride from human recombinant dopamine D2L receptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetD(2) dopamine receptor(Rat)
University of Pennsylvania

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 81993BDBM81993(Bromocriptine+ (GTP+) | BROMOCRIPTINE | Bromocript...)
Affinity DataKd:  17nMAssay Description:In vitro affinity at mutant D2 receptor (S194A) in C6 (glioma) cell membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetD(2) dopamine receptor(Human)
Neuroscience Research Centre

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 81993BDBM81993(Bromocriptine+ (GTP+) | BROMOCRIPTINE | Bromocript...)
Affinity DataKi:  19nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetD(2) dopamine receptor(Rat)
University of Pennsylvania

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 81993BDBM81993(Bromocriptine+ (GTP+) | BROMOCRIPTINE | Bromocript...)
Affinity DataKi:  54nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2011
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetD(2) dopamine receptor(Rat)
University of Pennsylvania

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 81993BDBM81993(Bromocriptine+ (GTP+) | BROMOCRIPTINE | Bromocript...)
Affinity DataKi:  68nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetD(2) dopamine receptor(Rat)
University of Pennsylvania

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 81993BDBM81993(Bromocriptine+ (GTP+) | BROMOCRIPTINE | Bromocript...)
Affinity DataKi:  83nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2011
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetD(2) dopamine receptor(Human)
Neuroscience Research Centre

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 81993BDBM81993(Bromocriptine+ (GTP+) | BROMOCRIPTINE | Bromocript...)
Affinity DataKi:  110nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)