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Found 247 with Last Name = 'boulouard' and Initial = 'm'
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Universite De Caen

US Patent
LigandPNGBDBM50079375(CHEMBL3417008 | US9663465, 20)
Affinity DataKi:  0.900nMAssay Description:Prior to these competition studies, a series of saturation curves were performed in order to check whether the pharmacological parameters Kd, Bmax an...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Cermn

Curated by ChEMBL
LigandPNGBDBM50079375(CHEMBL3417008 | US9663465, 20)
Affinity DataKi:  0.950nMAssay Description:Displacement of [3H]GR113808 from 5-HT4R in guinea pig brain membranes incubated for 30 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50106249(CHEMBL92139 | [2-(1-Benzenesulfonyl-1H-indol-4-yl)...)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]lysergic acid diethylamide from human 5-HT6 receptor transfected in HeLa cells after 60 mins by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Cermn

Curated by ChEMBL
LigandPNGBDBM50293279(1-Methyl-5-[(1-propylpiperidin-4-yl)methyloxy]-pyr...)
Affinity DataKi:  1.74nMAssay Description:Displacement of [3H]GR-113808 from 5HT4 receptor in guinea pig striatum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM21358(2-[1-({6-chloroimidazo[2,1-b][1,3]thiazole-5-}sulf...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]lysergic acid diethylamide from human 5-HT6 receptor expressed in HeLa cells after 120 mins by scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Cermn

Curated by ChEMBL
LigandPNGBDBM50558239(CHEMBL4781228)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-GR113808 from guinea pig brain 5HT4 receptor in presence of serotonin incubated for 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM34141(CHEMBL76237 | MS-245)
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]lysergic acid diethylamide from human 5-HT6 receptor transfected in HEK293 cells after 60 mins by liquid scintillation spectromet...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Cermn

Curated by ChEMBL
LigandPNGBDBM50079377(CHEMBL3417007)
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]GR113808 from 5-HT4R in guinea pig brain membranes incubated for 30 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Universite De Caen

US Patent
LigandPNGBDBM327460(4-amino-5-chloro-[[1-(cyclohexylmethyl)-4-piperidy...)
Affinity DataKi:  2.30nMAssay Description:Prior to these competition studies, a series of saturation curves were performed in order to check whether the pharmacological parameters Kd, Bmax an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Universite De Caen

US Patent
LigandPNGBDBM327466(1-[4-amino-5-chloro-2-(2-fluoroÚthoxy)phenyl]-3-[1...)
Affinity DataKi:  2.5nMAssay Description:Prior to these competition studies, a series of saturation curves were performed in order to check whether the pharmacological parameters Kd, Bmax an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Cermn

Curated by ChEMBL
LigandPNGBDBM50079367(CHEMBL3416998)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]GR113808 from 5-HT4R in guinea pig brain membranes incubated for 30 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Universite De Caen

US Patent
LigandPNGBDBM327456(1-(4-amino-5-chloro-2-methoxyphenyl)-3-[1-[(piperi...)
Affinity DataKi:  2.5nMAssay Description:Prior to these competition studies, a series of saturation curves were performed in order to check whether the pharmacological parameters Kd, Bmax an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50108392((3-ENDO)-8-METHYL-8-AZABICYCLO[3.2.1]OCT-3-YL 1H-I...)
Affinity DataKi:  2.80nMAssay Description:Binding affinity at 5HT3 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Cermn

Curated by ChEMBL
LigandPNGBDBM50122716(5-(Piperidin-4-ylmethoxy)-9-propyl-1,2,3,4-tetrahy...)
Affinity DataKi:  2.90nMAssay Description:Ability to displace [3H]GR-113808 from 5-hydroxytryptamine 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50106250(CHEMBL93868 | N,N-dimethyl-2-(1-(phenylsulfonyl)-1...)
Affinity DataKi:  2.90nMAssay Description:Displacement of [3H]lysergic acid diethylamide from human 5-HT6 receptor transfected in HeLa cells after 60 mins by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Universite De Caen

US Patent
LigandPNGBDBM50079365(CHEMBL3416996 | US9663465, 8)
Affinity DataKi:  3nMAssay Description:Prior to these competition studies, a series of saturation curves were performed in order to check whether the pharmacological parameters Kd, Bmax an...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Cermn

Curated by ChEMBL
LigandPNGBDBM50079365(CHEMBL3416996 | US9663465, 8)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]GR113808 from 5-HT4R in guinea pig brain membranes incubated for 30 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Normandie Univ

Curated by ChEMBL
LigandPNGBDBM28583(5-chloro-N-[4-methoxy-3-(piperazin-1-yl)phenyl]-3-...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in BHK cell membrane measured after 60 mins by scintillation counter methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Cermn

Curated by ChEMBL
LigandPNGBDBM50558245(CHEMBL4789661)
Affinity DataKi:  3.5nMAssay Description:Displacement of [3H]-GR113808 from guinea pig brain 5HT4 receptor in presence of serotonin incubated for 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Universite De Caen

US Patent
LigandPNGBDBM327448(1-(4-amino-5-fluoro-2-methoxyphenyl)-3-[1-(cyclohe...)
Affinity DataKi:  3.80nMAssay Description:Prior to these competition studies, a series of saturation curves were performed in order to check whether the pharmacological parameters Kd, Bmax an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Universite De Caen

US Patent
LigandPNGBDBM50079366(CHEMBL3416997 | US9663465, 12)
Affinity DataKi:  3.90nMAssay Description:Prior to these competition studies, a series of saturation curves were performed in order to check whether the pharmacological parameters Kd, Bmax an...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Cermn

Curated by ChEMBL
LigandPNGBDBM50079366(CHEMBL3416997 | US9663465, 12)
Affinity DataKi:  3.90nMAssay Description:Displacement of [3H]GR113808 from 5-HT4R in guinea pig brain membranes incubated for 30 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50562651(CHEMBL4788250)
Affinity DataKi:  4.30nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in HEK293 cell membrane measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50300828(2-(3-(3-fluorophenylsulfonyl)-1H-pyrrolo[2,3-b]pyr...)
Affinity DataKi:  4.80nMAssay Description:Displacement of [3H]lysergic acid diethylamide from human 5-HT6 receptor expressed in HeLa cells by scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Cermn

Curated by ChEMBL
LigandPNGBDBM50079369(CHEMBL3417000 | US9663465, 11)
Affinity DataKi:  4.90nMAssay Description:Displacement of [3H]GR113808 from 5-HT4R in guinea pig brain membranes incubated for 30 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Cermn

Curated by ChEMBL
LigandPNGBDBM50558234(CHEMBL4780536)
Affinity DataKi:  5.30nMAssay Description:Displacement of [3H]-GR113808 from guinea pig brain 5HT4 receptor in presence of serotonin incubated for 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Cermn

Curated by ChEMBL
LigandPNGBDBM50413548(CHEMBL512679)
Affinity DataKi:  5.37nMAssay Description:Displacement of [3H]GR-113808 from 5HT4 receptor in guinea pig striatum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Universite De Caen

US Patent
LigandPNGBDBM327461(4-amino-5-bromo-N-[[1-(cyclohexylmethyl)-4-piperid...)
Affinity DataKi:  5.40nMAssay Description:Prior to these competition studies, a series of saturation curves were performed in order to check whether the pharmacological parameters Kd, Bmax an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM21354(2-{1-[(5-chlorothiophene-2-)sulfonyl]-1H-indol-3-y...)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]lysergic acid diethylamide from human 5-HT6 receptor expressed in HeLa cells after 120 mins by scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Cermn

Curated by ChEMBL
LigandPNGBDBM50558243(CHEMBL4746550)
Affinity DataKi:  6.20nMAssay Description:Displacement of [3H]-GR113808 from guinea pig brain 5HT4 receptor in presence of serotonin incubated for 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Cermn

Curated by ChEMBL
LigandPNGBDBM50413547(CHEMBL448702)
Affinity DataKi:  6.46nMAssay Description:Displacement of [3H]GR-113808 from 5HT4 receptor in guinea pig striatum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Cermn

Curated by ChEMBL
LigandPNGBDBM50079362(CHEMBL3417009 | US9663465, 9)
Affinity DataKi:  6.60nMAssay Description:Displacement of [3H]GR113808 from 5-HT4R in guinea pig brain membranes incubated for 30 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50019754(IDALOPIRDINE | LU-AE58054)
Affinity DataKi:  6.90nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in HEK293 cell membrane measured after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Universite De Caen

US Patent
LigandPNGBDBM50079362(CHEMBL3417009 | US9663465, 9)
Affinity DataKi:  7.10nMAssay Description:Prior to these competition studies, a series of saturation curves were performed in order to check whether the pharmacological parameters Kd, Bmax an...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Cermn

Curated by ChEMBL
LigandPNGBDBM50558238(CHEMBL4741579)
Affinity DataKi:  7.70nMAssay Description:Displacement of [3H]-GR113808 from guinea pig brain 5HT4 receptor in presence of serotonin incubated for 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Universite De Caen

US Patent
LigandPNGBDBM50079369(CHEMBL3417000 | US9663465, 11)
Affinity DataKi:  8nMAssay Description:Prior to these competition studies, a series of saturation curves were performed in order to check whether the pharmacological parameters Kd, Bmax an...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Cermn

Curated by ChEMBL
LigandPNGBDBM50079368(CHEMBL3416999 | US9663465, 16)
Affinity DataKi:  8.20nMAssay Description:Displacement of [3H]GR113808 from 5-HT4R in guinea pig brain membranes incubated for 30 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Universite De Caen

US Patent
LigandPNGBDBM50079368(CHEMBL3416999 | US9663465, 16)
Affinity DataKi:  8.20nMAssay Description:Prior to these competition studies, a series of saturation curves were performed in order to check whether the pharmacological parameters Kd, Bmax an...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Cermn

Curated by ChEMBL
LigandPNGBDBM50558241(CHEMBL4760149)
Affinity DataKi:  8.20nMAssay Description:Displacement of [3H]-GR113808 from guinea pig brain 5HT4 receptor in presence of serotonin incubated for 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Cermn

Curated by ChEMBL
LigandPNGBDBM50413546(CHEMBL513254)
Affinity DataKi:  8.51nMAssay Description:Displacement of [3H]GR-113808 from 5HT4 receptor in guinea pig striatum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Cermn

Curated by ChEMBL
LigandPNGBDBM50558235(CHEMBL4799043)
Affinity DataKi:  8.70nMAssay Description:Displacement of [3H]-GR113808 from guinea pig brain 5HT4 receptor in presence of serotonin incubated for 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Cermn

Curated by ChEMBL
LigandPNGBDBM50413545(CHEMBL469575)
Affinity DataKi:  8.71nMAssay Description:Displacement of [3H]GR-113808 from 5HT4 receptor in guinea pig striatum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Cermn

Curated by ChEMBL
LigandPNGBDBM50079364(CHEMBL3416995 | US9663465, 7)
Affinity DataKi:  8.80nMAssay Description:Displacement of [3H]GR113808 from 5-HT4R in guinea pig brain membranes incubated for 30 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Universite De Caen

US Patent
LigandPNGBDBM50079364(CHEMBL3416995 | US9663465, 7)
Affinity DataKi:  8.80nMAssay Description:Prior to these competition studies, a series of saturation curves were performed in order to check whether the pharmacological parameters Kd, Bmax an...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Universite De Caen

US Patent
LigandPNGBDBM327445(1-(4-amino-5-bromo-2-methoxyphenyl)-3-[1-butyl-4-p...)
Affinity DataKi:  8.90nMAssay Description:Prior to these competition studies, a series of saturation curves were performed in order to check whether the pharmacological parameters Kd, Bmax an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Cermn

Curated by ChEMBL
LigandPNGBDBM84950(CAS_183782 | NSC_183782 | RS 67333)
Affinity DataKi:  9.30nMAssay Description:Displacement of [3H]GR113808 from 5-HT4R in guinea pig brain membranes incubated for 30 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Cermn

Curated by ChEMBL
LigandPNGBDBM50413544(CHEMBL511794)
Affinity DataKi:  9.55nMAssay Description:Displacement of [3H]GR-113808 from 5HT4 receptor in guinea pig striatum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Cermn

Curated by ChEMBL
LigandPNGBDBM50122722(9-Butyl-5-(piperidin-4-ylmethoxy)-1,2,3,4-tetrahyd...)
Affinity DataKi:  10nMAssay Description:Ability to displace [3H]GR-113808 from 5-hydroxytryptamine 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Cermn

Curated by ChEMBL
LigandPNGBDBM50122721(6-(1-Ethyl-piperidin-4-ylmethoxy)-8,9,10,11-tetrah...)
Affinity DataKi:  11nMAssay Description:Ability to displace [3H]GR-113808 from 5-hydroxytryptamine 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50562651(CHEMBL4788250)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in HEK293 cell membrane measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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