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Found 141 with Last Name = 'davis' and Initial = 'jr'
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50192169((R)-3,5-dimethoxy-N-(1-(naphthalen-2-ylmethyl)pyrr...)
Affinity DataKi:  7nMAssay Description:Binding activity against human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50192189(3,4,5-trifluoro-N-(1-(naphthalen-2-ylmethyl)piperi...)
Affinity DataKi:  9nMAssay Description:Binding activity against human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50168507((E)-N-(1-cinnamylpiperidin-4-yl)-3,5-dimethoxybenz...)
Affinity DataKi:  12nMAssay Description:Binding activity against human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50192178(3,5-dimethoxy-N-((3R)-1-(1-(naphthalen-2-yl)ethyl)...)
Affinity DataKi:  12nMAssay Description:Binding activity against human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50192174(4-fluoro-3-methoxy-N-(1-(naphthalen-2-ylmethyl)pip...)
Affinity DataKi:  13nMAssay Description:Binding activity against human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50192163((R,E)-N-(1-cinnamylpyrrolidin-3-yl)-3,5-dimethoxyb...)
Affinity DataKi:  17nMAssay Description:Binding activity against human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50192161(3,4-difluoro-N-(1-(naphthalen-2-ylmethyl)piperidin...)
Affinity DataKi:  18nMAssay Description:Binding activity against human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50192162(3,5-dimethoxy-N-((3R)-1-((E)-4-phenylbut-3-en-2-yl...)
Affinity DataKi:  23nMAssay Description:Binding activity against human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50192160(3,5-dimethoxy-N-(1-(1-(naphthalen-2-yl)ethyl)piper...)
Affinity DataKi:  25nMAssay Description:Binding activity against human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50192177(3,5-dimethoxy-N-(1-(naphthalen-2-ylmethyl)piperidi...)
Affinity DataKi:  27nMAssay Description:Binding activity against human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50192165(3-methoxy-N-(1-(naphthalen-2-ylmethyl)piperidin-4-...)
Affinity DataKi:  29nMAssay Description:Binding activity against human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50192182(CHEMBL214778 | N-(1-((6-fluoronaphthalen-2-yl)meth...)
Affinity DataKi:  32nMAssay Description:Binding activity against human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50192157(4-fluoro-N-(1-(naphthalen-2-ylmethyl)piperidin-4-y...)
Affinity DataKi:  36nMAssay Description:Binding activity against human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50192173((1R,5S,6r)-N-(3,4-difluorobenzyl)-3-(naphthalen-2-...)
Affinity DataKi:  40nMAssay Description:Binding activity against human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50192183(3,5-diethoxy-N-(1-(naphthalen-2-ylmethyl)piperidin...)
Affinity DataKi:  56nMAssay Description:Binding activity against human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50192168((R)-4-fluoro-3-methoxy-N-(1-(naphthalen-2-ylmethyl...)
Affinity DataKi:  62nMAssay Description:Binding activity against human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50192195(3,5-difluoro-N-(1-(naphthalen-2-ylmethyl)piperidin...)
Affinity DataKi:  65nMAssay Description:Binding activity against human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50192192((R)-3-methoxy-N-(1-(naphthalen-2-ylmethyl)pyrrolid...)
Affinity DataKi:  67nMAssay Description:Binding activity against human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50192164(3,5-dimethoxy-N-(4-methyl-1-(naphthalen-2-ylmethyl...)
Affinity DataKi:  86nMAssay Description:Binding activity against human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50241090(3,5-dimethoxy-N-(1-((6-methoxynaphthalen-2-yl)meth...)
Affinity DataKi:  99nMAssay Description:Binding activity against human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50192184(3-(dimethylamino)-N-(1-(naphthalen-2-ylmethyl)pipe...)
Affinity DataKi:  125nMAssay Description:Binding activity against human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50192167(CHEMBL214726 | N-(1-((6-fluoronaphthalen-2-yl)meth...)
Affinity DataKi:  125nMAssay Description:Binding activity against human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50192187(3,5-dimethoxy-N-((3R,4R)-3-methyl-1-(naphthalen-2-...)
Affinity DataKi:  133nMAssay Description:Binding activity against human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50192191(3,5-dimethoxy-N-(1-((1,2,3,4-tetrahydronaphthalen-...)
Affinity DataKi:  136nMAssay Description:Binding activity against human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50192170(3,5-dimethoxy-N-(1-((1-methyl-1H-indol-2-yl)methyl...)
Affinity DataKi:  142nMAssay Description:Binding activity against human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50192193(3,5-dimethoxy-N-methyl-N-(1-(naphthalen-2-ylmethyl...)
Affinity DataKi:  169nMAssay Description:Binding activity against human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50192186(3,5-dimethoxy-N-((3S,4R)-3-methyl-1-(naphthalen-2-...)
Affinity DataKi:  170nMAssay Description:Binding activity against human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50192159(CHEMBL385535 | N-(1-(3,4-dichlorobenzyl)piperidin-...)
Affinity DataKi:  205nMAssay Description:Binding activity against human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50192188(4-chloro-N-(1-(naphthalen-2-ylmethyl)piperidin-4-y...)
Affinity DataKi:  232nMAssay Description:Binding activity against human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50192166(3,4,5-trimethoxy-N-(1-(naphthalen-2-ylmethyl)piper...)
Affinity DataKi:  286nMAssay Description:Binding activity against human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50192158(CHEMBL214684 | N-(1-benzylpiperidin-4-yl)-3,5-dime...)
Affinity DataKi:  302nMAssay Description:Binding activity against human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50192179(CHEMBL215388 | N-(1-(naphthalen-2-ylmethyl)piperid...)
Affinity DataKi:  347nMAssay Description:Binding activity against human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50192194((S)-3,5-dimethoxy-N-(1-(naphthalen-2-ylmethyl)pyrr...)
Affinity DataKi:  484nMAssay Description:Binding activity against human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50192190((S)-N-(1-(3-hydroxy-3-phenylpropyl)piperidin-4-yl)...)
Affinity DataKi:  505nMAssay Description:Binding activity against human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50192181(3-hydroxy-N-(1-(naphthalen-2-ylmethyl)piperidin-4-...)
Affinity DataKi:  570nMAssay Description:Binding activity against human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50192172(3,5-dimethoxy-N-(1-(quinolin-2-ylmethyl)piperidin-...)
Affinity DataKi:  625nMAssay Description:Binding activity against human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50192171(3,4-dimethoxy-N-(1-(naphthalen-2-ylmethyl)piperidi...)
Affinity DataKi:  1.00E+3nMAssay Description:Binding activity against human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50192175((R)-N-(1-benzylpyrrolidin-3-yl)-3,5-dimethoxybenza...)
Affinity DataKi:  8.07E+3nMAssay Description:Binding activity against human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50192185((1R,5S,6s)-N-(3,4-difluorobenzyl)-3-(naphthalen-2-...)
Affinity DataKi: >1.00E+5nMAssay Description:Binding activity against human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50192180(3,5-dimethoxy-N-(2,2,6,6-tetramethyl-1-(naphthalen...)
Affinity DataKi: >1.00E+5nMAssay Description:Binding activity against human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50192156(3,5-dimethoxy-N-(1-(3-phenylpropyl)piperidin-4-yl)...)
Affinity DataKi: >1.00E+5nMAssay Description:Binding activity against human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50192176(3,5-dimethoxy-N-(3-(naphthalen-2-ylmethylamino)pro...)
Affinity DataKi: >1.00E+5nMAssay Description:Binding activity against human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50173041(3,5-dimethoxy-N-(1-(naphthalen-2-ylmethyl)piperidi...)
Affinity DataKi: >1.00E+5nMAssay Description:Binding activity against human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50193999(2-(3H-imidazo[4,5-c]pyridin-3-yl)-N-((S)-1-phenyle...)
Affinity DataIC50:  4nMAssay Description:Inhibition of JAK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50201514(2-(3H-imidazo[4,5-c]pyridin-3-yl)-N-methoxy-7-meth...)
Affinity DataIC50:  6nMAssay Description:Inhibition of JAK2 by kinase-Glo luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50194011(2-(3H-imidazo[4,5-c]pyridin-3-yl)-N4,N4-dimethyl-N...)
Affinity DataIC50:  7nMAssay Description:Inhibition of JAK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50193989(CHEMBL221976 | N-((S)-1-(4-fluorophenyl)ethyl)-2-(...)
Affinity DataIC50:  8nMAssay Description:Inhibition of JAK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50193995(3-((3R,4R)-4-methyl-3-(methyl(7H-pyrrolo[2,3-d]pyr...)
Affinity DataIC50:  11nMAssay Description:Inhibition of JAK2More data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50201503((2-(3H-imidazo[4,5-c]pyridin-3-yl)-7-methyl-4-((S)...)
Affinity DataIC50:  11nMAssay Description:Inhibition of JAK2 by kinase-Glo luminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50193995(3-((3R,4R)-4-methyl-3-(methyl(7H-pyrrolo[2,3-d]pyr...)
Affinity DataIC50:  11nMAssay Description:Inhibition of JAK2 by kinase-Glo luminescent assayMore data for this Ligand-Target Pair
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