Compile Data Set for Download or QSAR
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Found 103 with Last Name = 'fulco' and Initial = 'mc'
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Universit£ di Perugia

Curated by ChEMBL
LigandPNGBDBM17657((2S)-2-aminopentanedioic acid | (S)-Glu | D-Glutam...)
Affinity DataKi:  250nMAssay Description:Displacement of [3H]quisqualate from mGluR1 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Universit£ di Perugia

Curated by ChEMBL
LigandPNGBDBM17657((2S)-2-aminopentanedioic acid | (S)-Glu | D-Glutam...)
Affinity DataKi:  390nMAssay Description:Binding affinity to mGluR5 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
Universit£ di Perugia

Curated by ChEMBL
LigandPNGBDBM17657((2S)-2-aminopentanedioic acid | (S)-Glu | D-Glutam...)
Affinity DataKi:  2.40E+3nMAssay Description:Displacement of [3H]LAP4 from mGluR4 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Universit£ di Perugia

Curated by ChEMBL
LigandPNGBDBM17657((2S)-2-aminopentanedioic acid | (S)-Glu | D-Glutam...)
Affinity DataKi:  1.10E+4nMAssay Description:Displacement of [3H]LY341495 from mGluR2 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Universit£ di Perugia

Curated by ChEMBL
LigandPNGBDBM50220148((2S,1'R,2'S)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi:  3.40E+4nMAssay Description:Displacement of [3H]quisqualate from mGluR1 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Universit£ di Perugia

Curated by ChEMBL
LigandPNGBDBM50220148((2S,1'R,2'S)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi:  4.90E+4nMAssay Description:Binding affinity to mGluR5 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
Universit£ di Perugia

Curated by ChEMBL
LigandPNGBDBM50220147((S)-2-amino-4-sulfobutanoic acid | CHEMBL230951 | ...)
Affinity DataKi:  5.30E+4nMAssay Description:Displacement of [3H]LAP4 from mGluR4 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Universit£ di Perugia

Curated by ChEMBL
LigandPNGBDBM50220147((S)-2-amino-4-sulfobutanoic acid | CHEMBL230951 | ...)
Affinity DataKi:  5.40E+4nMAssay Description:Binding affinity to mGluR5 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Universit£ di Perugia

Curated by ChEMBL
LigandPNGBDBM50220154((2R,1'R,2'R)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi:  5.50E+4nMAssay Description:Binding affinity to mGluR5 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Universit£ di Perugia

Curated by ChEMBL
LigandPNGBDBM50220150((2R,1'S,2'R)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi:  6.70E+4nMAssay Description:Binding affinity to mGluR5 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Universit£ di Perugia

Curated by ChEMBL
LigandPNGBDBM50220149((2S,1'S,2'R)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi:  7.70E+4nMAssay Description:Displacement of [3H]quisqualate from mGluR1 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Universit£ di Perugia

Curated by ChEMBL
LigandPNGBDBM50220149((2S,1'S,2'R)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi:  8.10E+4nMAssay Description:Binding affinity to mGluR5 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Universit£ di Perugia

Curated by ChEMBL
LigandPNGBDBM50220147((S)-2-amino-4-sulfobutanoic acid | CHEMBL230951 | ...)
Affinity DataKi:  8.70E+4nMAssay Description:Displacement of [3H]quisqualate from mGluR1 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Universit£ di Perugia

Curated by ChEMBL
LigandPNGBDBM50220148((2S,1'R,2'S)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi:  2.35E+5nMAssay Description:Displacement of [3H]LY341495 from mGluR2 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Universit£ di Perugia

Curated by ChEMBL
LigandPNGBDBM50220150((2R,1'S,2'R)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi:  2.54E+5nMAssay Description:Displacement of [3H]quisqualate from mGluR1 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Universit£ di Perugia

Curated by ChEMBL
LigandPNGBDBM50220154((2R,1'R,2'R)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi: >3.00E+5nMAssay Description:Displacement of [3H]quisqualate from mGluR1 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Universit£ di Perugia

Curated by ChEMBL
LigandPNGBDBM50220151((2R,1'S,2'S)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi: >3.00E+5nMAssay Description:Displacement of [3H]LY341495 from mGluR2 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Universit£ di Perugia

Curated by ChEMBL
LigandPNGBDBM50220151((2R,1'S,2'S)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi: >3.00E+5nMAssay Description:Displacement of [3H]quisqualate from mGluR1 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Universit£ di Perugia

Curated by ChEMBL
LigandPNGBDBM50220153((2R,1'R,2'S)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi: >3.00E+5nMAssay Description:Displacement of [3H]quisqualate from mGluR1 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
Universit£ di Perugia

Curated by ChEMBL
LigandPNGBDBM50220148((2S,1'R,2'S)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi: >3.00E+5nMAssay Description:Displacement of [3H]LAP4 from mGluR4 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Universit£ di Perugia

Curated by ChEMBL
LigandPNGBDBM50220153((2R,1'R,2'S)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi: >3.00E+5nMAssay Description:Binding affinity to mGluR5 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
Universit£ di Perugia

Curated by ChEMBL
LigandPNGBDBM50220145((2S,1'R,2'R)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi: >3.00E+5nMAssay Description:Displacement of [3H]LAP4 from mGluR4 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
Universit£ di Perugia

Curated by ChEMBL
LigandPNGBDBM50220146((2S,1'S,2'S)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi: >3.00E+5nMAssay Description:Displacement of [3H]LAP4 from mGluR4 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
Universit£ di Perugia

Curated by ChEMBL
LigandPNGBDBM50220154((2R,1'R,2'R)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi: >3.00E+5nMAssay Description:Displacement of [3H]LAP4 from mGluR4 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Universit£ di Perugia

Curated by ChEMBL
LigandPNGBDBM50220153((2R,1'R,2'S)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi: >3.00E+5nMAssay Description:Displacement of [3H]LY341495 from mGluR2 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Universit£ di Perugia

Curated by ChEMBL
LigandPNGBDBM50220151((2R,1'S,2'S)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi: >3.00E+5nMAssay Description:Binding affinity to mGluR5 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Universit£ di Perugia

Curated by ChEMBL
LigandPNGBDBM50220146((2S,1'S,2'S)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi: >3.00E+5nMAssay Description:Displacement of [3H]quisqualate from mGluR1 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Universit£ di Perugia

Curated by ChEMBL
LigandPNGBDBM50220145((2S,1'R,2'R)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi: >3.00E+5nMAssay Description:Displacement of [3H]LY341495 from mGluR2 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Universit£ di Perugia

Curated by ChEMBL
LigandPNGBDBM50220146((2S,1'S,2'S)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi: >3.00E+5nMAssay Description:Displacement of [3H]LY341495 from mGluR2 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Universit£ di Perugia

Curated by ChEMBL
LigandPNGBDBM50220150((2R,1'S,2'R)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi: >3.00E+5nMAssay Description:Displacement of [3H]LY341495 from mGluR2 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Universit£ di Perugia

Curated by ChEMBL
LigandPNGBDBM50220149((2S,1'S,2'R)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi: >3.00E+5nMAssay Description:Displacement of [3H]LY341495 from mGluR2 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Universit£ di Perugia

Curated by ChEMBL
LigandPNGBDBM50220145((2S,1'R,2'R)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi: >3.00E+5nMAssay Description:Binding affinity to mGluR5 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
Universit£ di Perugia

Curated by ChEMBL
LigandPNGBDBM50220153((2R,1'R,2'S)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi: >3.00E+5nMAssay Description:Displacement of [3H]LAP4 from mGluR4 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
Universit£ di Perugia

Curated by ChEMBL
LigandPNGBDBM50220150((2R,1'S,2'R)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi: >3.00E+5nMAssay Description:Displacement of [3H]LAP4 from mGluR4 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Universit£ di Perugia

Curated by ChEMBL
LigandPNGBDBM50220145((2S,1'R,2'R)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi: >3.00E+5nMAssay Description:Displacement of [3H]quisqualate from mGluR1 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Universit£ di Perugia

Curated by ChEMBL
LigandPNGBDBM50220146((2S,1'S,2'S)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi: >3.00E+5nMAssay Description:Binding affinity to mGluR5 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Universit£ di Perugia

Curated by ChEMBL
LigandPNGBDBM50220147((S)-2-amino-4-sulfobutanoic acid | CHEMBL230951 | ...)
Affinity DataKi: >3.00E+5nMAssay Description:Displacement of [3H]LY341495 from mGluR2 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
Universit£ di Perugia

Curated by ChEMBL
LigandPNGBDBM50220149((2S,1'S,2'R)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi: >3.00E+5nMAssay Description:Displacement of [3H]LAP4 from mGluR4 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Universit£ di Perugia

Curated by ChEMBL
LigandPNGBDBM50220154((2R,1'R,2'R)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi: >3.00E+5nMAssay Description:Displacement of [3H]LY341495 from mGluR2 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
Universit£ di Perugia

Curated by ChEMBL
LigandPNGBDBM50220151((2R,1'S,2'S)-2-(2'-sulfonocyclopropyl)glycine | CH...)
Affinity DataKi: >3.00E+5nMAssay Description:Displacement of [3H]LAP4 from mGluR4 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
European Institute of Oncology

Curated by ChEMBL
LigandPNGBDBM50141381(CHEMBL3758184)
Affinity DataIC50:  1nMAssay Description:Inhibition of HDAC in human HeLa cells nuclear extract using Fluor de lys as substrate after 15 mins by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
DAC SRL

Curated by ChEMBL
LigandPNGBDBM50361444(CHEMBL1938433)
Affinity DataIC50:  9.40nMAssay Description:Inhibition of HDAC3 using carboxyfluorescein-labeled peptide as substrate after 17 hrs by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
DAC SRL

Curated by ChEMBL
LigandPNGBDBM50361444(CHEMBL1938433)
Affinity DataIC50:  25.7nMAssay Description:Inhibition of HDAC6 using carboxyfluorescein-labeled peptide as substrate after 17 hrs by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
European Institute of Oncology

Curated by ChEMBL
LigandPNGBDBM50141111(CHEMBL3758901)
Affinity DataIC50:  26nMAssay Description:Inhibition of HDAC in human HeLa cells nuclear extract using Fluor de lys as substrate after 15 mins by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
European Institute of Oncology

Curated by ChEMBL
LigandPNGBDBM50141185(CHEMBL3759550)
Affinity DataIC50:  27nMAssay Description:Inhibition of HDAC in human HeLa cells nuclear extract using Fluor de lys as substrate after 15 mins by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
DAC SRL

Curated by ChEMBL
LigandPNGBDBM50141111(CHEMBL3758901)
Affinity DataIC50:  28nMAssay Description:Inhibition of HDAC3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
DAC SRL

Curated by ChEMBL
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)
Affinity DataIC50:  29nMAssay Description:Inhibition of HDAC6 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetHistone deacetylase 3(Homo sapiens (Human))
DAC SRL

Curated by ChEMBL
LigandPNGBDBM50141139(CHEMBL3759808)
Affinity DataIC50:  30nMAssay Description:Inhibition of HDAC3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
European Institute of Oncology

Curated by ChEMBL
LigandPNGBDBM50141361(CHEMBL3758716)
Affinity DataIC50:  34nMAssay Description:Inhibition of HDAC in human HeLa cells nuclear extract using Fluor de lys as substrate after 15 mins by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
European Institute of Oncology

Curated by ChEMBL
LigandPNGBDBM50141111(CHEMBL3758901)
Affinity DataIC50:  52nMAssay Description:Inhibition of HDAC in human HeLa cells nuclear extract using Fluor de lys as substrate after 15 mins by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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