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Found 60 with Last Name = 'hernandes' and Initial = 'mz'
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universidade Federal de Pernambuco

Curated by ChEMBL
LigandPNGBDBM50320887(3-(2-Chloro-6-fluoro-benzyl)-5-(2,4-dichlorobenzyl...)
Affinity DataKi:  4.00E+3nMAssay Description:Displacement of [3H]rosiglitazone from human PPARgamma ligand binding domain expressed in Escherichia coli BL21 after 12 hrs by liquid scintillation ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universidade Federal de Pernambuco

Curated by ChEMBL
LigandPNGBDBM50320886(3-(2-Bromo-benzyl)-5-(4-methanesulfonyl-benzyliden...)
Affinity DataKi:  7.30E+3nMAssay Description:Displacement of [3H]rosiglitazone from human PPARgamma ligand binding domain expressed in Escherichia coli BL21 after 12 hrs by liquid scintillation ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universidade Federal de Pernambuco

Curated by ChEMBL
LigandPNGBDBM50320884(3-(3-Chloro-benzyl)-5-(4-methanesulfonyl-benzylide...)
Affinity DataKi:  4.30E+4nMAssay Description:Displacement of [3H]rosiglitazone from human PPARgamma ligand binding domain expressed in Escherichia coli BL21 after 12 hrs by liquid scintillation ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universidade Federal de Pernambuco

Curated by ChEMBL
LigandPNGBDBM50320885(5-Bipheny-4-ylmethylene-3-(3-chloro-benzyl)-thiazo...)
Affinity DataKi:  4.36E+4nMAssay Description:Displacement of [3H]rosiglitazone from human PPARgamma ligand binding domain expressed in Escherichia coli BL21 after 12 hrs by liquid scintillation ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Universidade Federal de Pernambuco

Curated by ChEMBL
LigandPNGBDBM50058809(CHEMBL3329524)
Affinity DataIC50:  10nMAssay Description:Inhibition of recombinant Trypanosoma cruzi cruzain using Z-Phe-Argaminomethylcoumarin as fluorogenic substrate preincubated for 10 mins before subst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Universidade Federal de Pernambuco

Curated by ChEMBL
LigandPNGBDBM50058806(CHEMBL3329519)
Affinity DataIC50:  40nMAssay Description:Inhibition of recombinant Trypanosoma cruzi cruzain using Z-Phe-Argaminomethylcoumarin as fluorogenic substrate preincubated for 10 mins before subst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Universidade Federal de Pernambuco

Curated by ChEMBL
LigandPNGBDBM50114613((1E)-1-(3-bromophenyl)propan-1-one thiosemicarbazo...)
Affinity DataIC50:  40nMAssay Description:Inhibition of recombinant Trypanosoma cruzi cruzain using Z-FR-AMC as substrate and measured at 12 sec interval for 5 mins by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Universidade Federal de Pernambuco

Curated by ChEMBL
LigandPNGBDBM50114613((1E)-1-(3-bromophenyl)propan-1-one thiosemicarbazo...)
Affinity DataIC50:  40nMAssay Description:Inhibition of Trypanosoma cruzi cruzaine pre-incubated for 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Universidade Federal de Pernambuco

Curated by ChEMBL
LigandPNGBDBM50330929(2-[(p-Methylphenyl)thiopropylidenehydrazinyl]-5-me...)
Affinity DataIC50:  60nMAssay Description:Inhibition of Trypanosoma cruzi cruzaine pre-incubated for 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Universidade Federal de Pernambuco

Curated by ChEMBL
LigandPNGBDBM50114653((1E)-1-(3,4-dichlorophenyl)ethan-1-one thiosemicar...)
Affinity DataIC50:  100nMAssay Description:Inhibition of Trypanosoma cruzi cruzaine pre-incubated for 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Universidade Federal de Pernambuco

Curated by ChEMBL
LigandPNGBDBM50330926(2-[(p-Chlorophenylthio)propylide-1-enehydrazinyl]-...)
Affinity DataIC50:  200nMAssay Description:Inhibition of Trypanosoma cruzi cruzaine pre-incubated for 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Universidade Federal de Pernambuco

Curated by ChEMBL
LigandPNGBDBM50058805(CHEMBL3329518)
Affinity DataIC50:  300nMAssay Description:Inhibition of recombinant Trypanosoma cruzi cruzain using Z-Phe-Argaminomethylcoumarin as fluorogenic substrate preincubated for 10 mins before subst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Universidade Federal de Pernambuco

Curated by ChEMBL
LigandPNGBDBM50058804(CHEMBL3329515)
Affinity DataIC50:  400nMAssay Description:Inhibition of recombinant Trypanosoma cruzi cruzain using Z-Phe-Argaminomethylcoumarin as fluorogenic substrate preincubated for 10 mins before subst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Universidade Federal de Pernambuco

Curated by ChEMBL
LigandPNGBDBM50330928(2-[(Phenylthio)propylide-1-enehydrazinyl]-5-methyl...)
Affinity DataIC50:  400nMAssay Description:Inhibition of Trypanosoma cruzi recombinant cruzain using Z-FR-AMC as substrate preincubated for 10 mins before substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Universidade Federal de Pernambuco

Curated by ChEMBL
LigandPNGBDBM50330928(2-[(Phenylthio)propylide-1-enehydrazinyl]-5-methyl...)
Affinity DataIC50:  400nMAssay Description:Inhibition of Trypanosoma cruzi cruzaine pre-incubated for 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Universidade Federal de Pernambuco

Curated by ChEMBL
LigandPNGBDBM50058808(CHEMBL3329521)
Affinity DataIC50:  400nMAssay Description:Inhibition of recombinant Trypanosoma cruzi cruzain using Z-Phe-Argaminomethylcoumarin as fluorogenic substrate preincubated for 10 mins before subst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Universidade Federal de Pernambuco

Curated by ChEMBL
LigandPNGBDBM50558296(CHEMBL4744510)
Affinity DataIC50:  510nMAssay Description:Inhibition of recombinant Trypanosoma cruzi cruzain using Z-FR-AMC as substrate and measured at 12 sec interval for 5 mins by fluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Universidade Federal de Pernambuco

Curated by ChEMBL
LigandPNGBDBM50058803(CHEMBL2409542)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of recombinant Trypanosoma cruzi cruzain using Z-Phe-Argaminomethylcoumarin as fluorogenic substrate preincubated for 10 mins before subst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Universidade Federal de Pernambuco

Curated by ChEMBL
LigandPNGBDBM50058802(CHEMBL3329513)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of recombinant Trypanosoma cruzi cruzain using Z-Phe-Argaminomethylcoumarin as fluorogenic substrate preincubated for 10 mins before subst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Universidade Federal de Pernambuco

Curated by ChEMBL
LigandPNGBDBM50558297(CHEMBL3787543)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibition of recombinant Trypanosoma cruzi cruzain using Z-FR-AMC as substrate and measured at 12 sec interval for 5 mins by fluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Universidade Federal de Pernambuco

Curated by ChEMBL
LigandPNGBDBM50058807(CHEMBL3329520)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibition of recombinant Trypanosoma cruzi cruzain using Z-Phe-Argaminomethylcoumarin as fluorogenic substrate preincubated for 10 mins before subst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Universidade Federal de Pernambuco

Curated by ChEMBL
LigandPNGBDBM50400185(CHEMBL2180342)
Affinity DataIC50:  6.60E+3nMAssay Description:Inhibition of Trypanosoma cruzi recombinant cruzain using Z-FR-AMC as substrate preincubated for 10 mins before substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Universidade Federal de Pernambuco

Curated by ChEMBL
LigandPNGBDBM50400195(CHEMBL2180344)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of Trypanosoma cruzi recombinant cruzain using Z-FR-AMC as substrate preincubated for 10 mins before substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Universidade Federal de Pernambuco

Curated by ChEMBL
LigandPNGBDBM50400188(CHEMBL2180670)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of Trypanosoma cruzi recombinant cruzain using Z-FR-AMC as substrate preincubated for 10 mins before substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Universidade Federal de Pernambuco

Curated by ChEMBL
LigandPNGBDBM50400197(CHEMBL2180347)
Affinity DataIC50:  8.70E+3nMAssay Description:Inhibition of Trypanosoma cruzi recombinant cruzain using Z-FR-AMC as substrate preincubated for 10 mins before substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Universidade Federal de Pernambuco

Curated by ChEMBL
LigandPNGBDBM50058801(CHEMBL3329506)
Affinity DataIC50:  9.50E+3nMAssay Description:Inhibition of recombinant Trypanosoma cruzi cruzain using Z-Phe-Argaminomethylcoumarin as fluorogenic substrate preincubated for 10 mins before subst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Universidade Federal de Pernambuco

Curated by ChEMBL
LigandPNGBDBM50558295(CHEMBL4782594)
Affinity DataIC50:  9.50E+3nMAssay Description:Inhibition of recombinant Trypanosoma cruzi cruzain using Z-FR-AMC as substrate and measured at 12 sec interval for 5 mins by fluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Universidade Federal de Pernambuco

Curated by ChEMBL
LigandPNGBDBM50400186(CHEMBL2180341)
Affinity DataIC50:  9.50E+3nMAssay Description:Inhibition of Trypanosoma cruzi recombinant cruzain using Z-FR-AMC as substrate preincubated for 10 mins before substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Universidade Federal de Pernambuco

Curated by ChEMBL
LigandPNGBDBM50400187(CHEMBL2180339)
Affinity DataIC50:  1.02E+4nMAssay Description:Inhibition of Trypanosoma cruzi recombinant cruzain using Z-FR-AMC as substrate preincubated for 10 mins before substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Universidade Federal de Pernambuco

Curated by ChEMBL
LigandPNGBDBM50400196(CHEMBL2180340)
Affinity DataIC50:  1.08E+4nMAssay Description:Inhibition of Trypanosoma cruzi recombinant cruzain using Z-FR-AMC as substrate preincubated for 10 mins before substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Universidade Federal de Pernambuco

Curated by ChEMBL
LigandPNGBDBM50400195(CHEMBL2180344)
Affinity DataIC50:  1.08E+4nMAssay Description:Inhibition of recombinant cathepsin L using ZFR-pNA as substrate preincubated for 45 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Universidade Federal de Pernambuco

Curated by ChEMBL
LigandPNGBDBM50558293(CHEMBL4747507)
Affinity DataIC50:  1.13E+4nMAssay Description:Inhibition of recombinant Trypanosoma cruzi cruzain using Z-FR-AMC as substrate and measured at 12 sec interval for 5 mins by fluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Universidade Federal de Pernambuco

Curated by ChEMBL
LigandPNGBDBM50400194(CHEMBL2180346)
Affinity DataIC50:  1.18E+4nMAssay Description:Inhibition of Trypanosoma cruzi recombinant cruzain using Z-FR-AMC as substrate preincubated for 10 mins before substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Universidade Federal de Pernambuco

Curated by ChEMBL
LigandPNGBDBM50400193(CHEMBL2180345)
Affinity DataIC50:  1.38E+4nMAssay Description:Inhibition of recombinant cathepsin L using ZFR-pNA as substrate preincubated for 45 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Universidade Federal de Pernambuco

Curated by ChEMBL
LigandPNGBDBM50558292(CHEMBL3787688)
Affinity DataIC50:  1.46E+4nMAssay Description:Inhibition of recombinant Trypanosoma cruzi cruzain using Z-FR-AMC as substrate and measured at 12 sec interval for 5 mins by fluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Universidade Federal de Pernambuco

Curated by ChEMBL
LigandPNGBDBM50558294(CHEMBL4746565)
Affinity DataIC50:  1.51E+4nMAssay Description:Inhibition of recombinant Trypanosoma cruzi cruzain using Z-FR-AMC as substrate and measured at 12 sec interval for 5 mins by fluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Universidade Federal de Pernambuco

Curated by ChEMBL
LigandPNGBDBM50558290(CHEMBL4744489)
Affinity DataIC50:  1.65E+4nMAssay Description:Inhibition of recombinant Trypanosoma cruzi cruzain using Z-FR-AMC as substrate and measured at 12 sec interval for 5 mins by fluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Universidade Federal de Pernambuco

Curated by ChEMBL
LigandPNGBDBM50400193(CHEMBL2180345)
Affinity DataIC50:  1.87E+4nMAssay Description:Inhibition of Trypanosoma cruzi recombinant cruzain using Z-FR-AMC as substrate preincubated for 10 mins before substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Universidade Federal de Pernambuco

Curated by ChEMBL
LigandPNGBDBM50400192(CHEMBL2180665)
Affinity DataIC50:  1.89E+4nMAssay Description:Inhibition of Trypanosoma cruzi recombinant cruzain using Z-FR-AMC as substrate preincubated for 10 mins before substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Universidade Federal de Pernambuco

Curated by ChEMBL
LigandPNGBDBM50558289(CHEMBL3785603)
Affinity DataIC50:  1.92E+4nMAssay Description:Inhibition of recombinant Trypanosoma cruzi cruzain using Z-FR-AMC as substrate and measured at 12 sec interval for 5 mins by fluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Universidade Federal de Pernambuco

Curated by ChEMBL
LigandPNGBDBM50400191(CHEMBL2180349)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of Trypanosoma cruzi recombinant cruzain using Z-FR-AMC as substrate at 20 uM preincubated for 10 mins before substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Universidade Federal de Pernambuco

Curated by ChEMBL
LigandPNGBDBM50330927(2-[(p-Methylphenylthio)ethylidenehydrazinyl]-5-met...)
Affinity DataIC50:  2.04E+4nMAssay Description:Inhibition of Trypanosoma cruzi recombinant cruzain using Z-FR-AMC as substrate preincubated for 10 mins before substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Universidade Federal de Pernambuco

Curated by ChEMBL
LigandPNGBDBM50330927(2-[(p-Methylphenylthio)ethylidenehydrazinyl]-5-met...)
Affinity DataIC50:  2.04E+4nMAssay Description:Inhibition of Trypanosoma cruzi cruzaine pre-incubated for 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Universidade Federal de Pernambuco

Curated by ChEMBL
LigandPNGBDBM50400189(CHEMBL2180669)
Affinity DataIC50:  3.19E+4nMAssay Description:Inhibition of Trypanosoma cruzi recombinant cruzain using Z-FR-AMC as substrate preincubated for 10 mins before substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Universidade Federal de Pernambuco

Curated by ChEMBL
LigandPNGBDBM50558291(CHEMBL4743580)
Affinity DataIC50:  3.27E+4nMAssay Description:Inhibition of recombinant Trypanosoma cruzi cruzain using Z-FR-AMC as substrate and measured at 12 sec interval for 5 mins by fluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Universidade Federal de Pernambuco

Curated by ChEMBL
LigandPNGBDBM50558288(CHEMBL3785430)
Affinity DataIC50:  4.46E+4nMAssay Description:Inhibition of recombinant Trypanosoma cruzi cruzain using Z-FR-AMC as substrate and measured at 12 sec interval for 5 mins by fluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Universidade Federal de Pernambuco

Curated by ChEMBL
LigandPNGBDBM50400185(CHEMBL2180342)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant cathepsin S using ZFR-pNA as substrate preincubated for 45 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Universidade Federal de Pernambuco

Curated by ChEMBL
LigandPNGBDBM50400186(CHEMBL2180341)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant cathepsin S using ZFR-pNA as substrate preincubated for 45 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Universidade Federal de Pernambuco

Curated by ChEMBL
LigandPNGBDBM50400187(CHEMBL2180339)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant cathepsin S using ZFR-pNA as substrate preincubated for 45 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Universidade Federal de Pernambuco

Curated by ChEMBL
LigandPNGBDBM50400188(CHEMBL2180670)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant cathepsin S using ZFR-pNA as substrate preincubated for 45 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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