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Found 812 with Last Name = 'peng' and Initial = 'b'
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50433602(CHEMBL2381980)
Affinity DataKi:  0.720nMAssay Description:Competitive inhibition of JAK2 (unknown origin)More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec Inc

Curated by ChEMBL
LigandPNGBDBM21190(4-(2-{[5-amino-2-(furan-2-yl)-[1,2,4]triazolo[1,5-...)
Affinity DataKi:  0.900nMAssay Description:Inhibition of [3H]-ZM-241,385 binidng to rat brain adenosine A2a receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec Inc

Curated by ChEMBL
LigandPNGBDBM21190(4-(2-{[5-amino-2-(furan-2-yl)-[1,2,4]triazolo[1,5-...)
Affinity DataKi:  0.900nMAssay Description:Inhibition of [3H]ZM-241385 binding to adenosine A2a receptor of rat brain tissueMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50433601(CHEMBL2381983)
Affinity DataKi:  1.40nMAssay Description:Competitive inhibition of JAK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec Inc

Curated by ChEMBL
LigandPNGBDBM50163407(2-Furan-2-yl-N*5*-[(R)-1-(2,4,6-trifluoro-benzyl)-...)
Affinity DataKi:  2nMAssay Description:Inhibition of [3H]ZM-241385 binding to adenosine A2a receptor of rat brain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec Inc

Curated by ChEMBL
LigandPNGBDBM50151189(5-[4-(3,5-Dichloro-pyridin-4-ylmethyl)-piperazin-1...)
Affinity DataKi:  2nMAssay Description:Inhibition of [3H]-ZM-241,385 binidng to rat brain adenosine A2a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec Inc

Curated by ChEMBL
LigandPNGBDBM50151182(2-Furan-2-yl-5-[4-(2,4,6-trifluoro-benzyl)-piperaz...)
Affinity DataKi:  3nMAssay Description:Inhibition of [3H]-ZM-241,385 binidng to rat brain adenosine A2a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec Inc

Curated by ChEMBL
LigandPNGBDBM50163432(CHEMBL179478 | N*5*-[(R)-1-(5-Chloro-furan-2-ylmet...)
Affinity DataKi:  3nMAssay Description:Inhibition of [3H]ZM-241385 binding to adenosine A2a receptor of rat brain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec Inc

Curated by ChEMBL
LigandPNGBDBM50151182(2-Furan-2-yl-5-[4-(2,4,6-trifluoro-benzyl)-piperaz...)
Affinity DataKi:  3nMAssay Description:Binding affinity against Adenosine A2a receptor determined using [3H]-ZM-241,385 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec Inc

Curated by ChEMBL
LigandPNGBDBM50151182(2-Furan-2-yl-5-[4-(2,4,6-trifluoro-benzyl)-piperaz...)
Affinity DataKi:  3nMAssay Description:Inhibition of [3H]ZM-241385 binding to adenosine A2a receptor of rat brain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec Inc

Curated by ChEMBL
LigandPNGBDBM50163423(2-Furan-2-yl-N*5*-[(R)-1-(2,3,6-trifluoro-benzyl)-...)
Affinity DataKi:  4nMAssay Description:Inhibition of [3H]ZM-241385 binding to adenosine A2a receptor of rat brain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec Inc

Curated by ChEMBL
LigandPNGBDBM50152215(7N-[1-(2-chloro-4-pyridylmethyl)-(2R)-tetrahydro-1...)
Affinity DataKi:  4nMAssay Description:Inhibition of [3H]ZM-241385 binding to adenosine A2a receptor of rat brain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec Inc

Curated by ChEMBL
LigandPNGBDBM50152215(7N-[1-(2-chloro-4-pyridylmethyl)-(2R)-tetrahydro-1...)
Affinity DataKi:  4nMAssay Description:Binding affinity against Adenosine A2a receptor from rat brain tissue was determined using [3H]-ZM-241,385 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec Inc

Curated by ChEMBL
LigandPNGBDBM50163402(CHEMBL176071 | N*5*-[(R)-1-(2-Fluoro-5-trifluorome...)
Affinity DataKi:  4nMAssay Description:Inhibition of [3H]ZM-241385 binding to adenosine A2a receptor of rat brain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec Inc

Curated by ChEMBL
LigandPNGBDBM50152240(CHEMBL184309 | N*5*-{2-[4-(2,4-Difluoro-phenyl)-pi...)
Affinity DataKi:  4nMAssay Description:Binding affinity against Adenosine A2a receptor determined using [3H]-ZM-241,385 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec Inc

Curated by ChEMBL
LigandPNGBDBM50163404(CHEMBL177615 | N*5*-[(R)-1-(2-Chloro-3,6-difluoro-...)
Affinity DataKi:  4nMAssay Description:Inhibition of [3H]ZM-241385 binding to adenosine A2a receptor of rat brain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec Inc

Curated by ChEMBL
LigandPNGBDBM50156604(CHEMBL173672 | N*5*-[(R)-1-(2,6-Difluoro-benzyl)-p...)
Affinity DataKi:  4nMAssay Description:Inhibition of [3H]ZM-241385 binding to adenosine A2a receptor of rat brain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec Inc

Curated by ChEMBL
LigandPNGBDBM50163422(CHEMBL368201 | N*5*-[(R)-1-(2-Fluoro-4-trifluorome...)
Affinity DataKi:  5nMAssay Description:Inhibition of [3H]ZM-241385 binding to adenosine A2a receptor of rat brain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec Inc

Curated by ChEMBL
LigandPNGBDBM50163420(CHEMBL177532 | N*5*-[(R)-1-(2,3-Difluoro-benzyl)-p...)
Affinity DataKi:  5nMAssay Description:Inhibition of [3H]ZM-241385 binding to adenosine A2a receptor of rat brain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec Inc

Curated by ChEMBL
LigandPNGBDBM50151186(5-[4-(6-Chloro-2,3-difluoro-benzyl)-piperazin-1-yl...)
Affinity DataKi:  5nMAssay Description:Inhibition of [3H]-ZM-241,385 binidng to rat brain adenosine A2a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec Inc

Curated by ChEMBL
LigandPNGBDBM50152222(CHEMBL360840 | N*5*-[(R)-1-(2-Fluoro-benzyl)-pyrro...)
Affinity DataKi:  6nMAssay Description:Binding affinity against Adenosine A2a receptor from rat brain tissue was determined using [3H]-ZM-241,385 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec Inc

Curated by ChEMBL
LigandPNGBDBM50151171(5-[4-(2-Chloro-quinolin-3-ylmethyl)-piperazin-1-yl...)
Affinity DataKi:  6nMAssay Description:Inhibition of [3H]-ZM-241,385 binidng to rat brain adenosine A2a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec Inc

Curated by ChEMBL
LigandPNGBDBM50152233(CHEMBL363660 | N*7*-{2-[4-(2,4-Difluoro-phenyl)-pi...)
Affinity DataKi:  6.5nMAssay Description:Binding affinity against Adenosine A2a receptor determined using [3H]-ZM-241,385 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec Inc

Curated by ChEMBL
LigandPNGBDBM50163425(2-Furan-2-yl-N*5*-((R)-1-pyridin-3-ylmethyl-pyrrol...)
Affinity DataKi:  7nMAssay Description:Inhibition of [3H]ZM-241385 binding to adenosine A2a receptor of rat brain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec Inc

Curated by ChEMBL
LigandPNGBDBM50163401(CHEMBL369373 | N*5*-[(R)-1-(3-Chloro-1-methyl-1H-p...)
Affinity DataKi:  7nMAssay Description:Inhibition of [3H]ZM-241385 binding to adenosine A2a receptor of rat brain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec Inc

Curated by ChEMBL
LigandPNGBDBM50163410(CHEMBL173993 | N*5*-[(R)-1-(3-Chloro-2-fluoro-benz...)
Affinity DataKi:  7nMAssay Description:Inhibition of [3H]ZM-241385 binding to adenosine A2a receptor of rat brain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec Inc

Curated by ChEMBL
LigandPNGBDBM50152234(CHEMBL184061 | N*5*-{2-[4-(2,4-Difluoro-phenyl)-pi...)
Affinity DataKi:  7.10nMAssay Description:Binding affinity against Adenosine A2a receptor determined using [3H]-ZM-241,385 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec Inc

Curated by ChEMBL
LigandPNGBDBM50163412(2-Furan-2-yl-N*5*-[(R)-1-(2,4,5-trifluoro-benzyl)-...)
Affinity DataKi:  8nMAssay Description:Inhibition of [3H]ZM-241385 binding to adenosine A2a receptor of rat brain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec Inc

Curated by ChEMBL
LigandPNGBDBM50163396(CHEMBL367593 | N*5*-[(R)-1-(3-Chloro-2-fluoro-6-tr...)
Affinity DataKi:  8nMAssay Description:Inhibition of [3H]ZM-241385 binding to adenosine A2a receptor of rat brain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec Inc

Curated by ChEMBL
LigandPNGBDBM50152220(CHEMBL183531 | N*7*-[(R)-1-(2-Chloro-pyridin-4-ylm...)
Affinity DataKi:  10nMAssay Description:Binding affinity against Adenosine A2a receptor from rat brain tissue was determined using [3H]-ZM-241,385 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec Inc

Curated by ChEMBL
LigandPNGBDBM50151181(2-Furan-2-yl-5-[4-(2,3,6-trifluoro-benzyl)-piperaz...)
Affinity DataKi:  10nMAssay Description:Inhibition of [3H]-ZM-241,385 binidng to rat brain adenosine A2a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec Inc

Curated by ChEMBL
LigandPNGBDBM50152214(2-Furan-2-yl-N*5*-methyl-N*5*-[(R)-1-(5-methyl-iso...)
Affinity DataKi:  11nMAssay Description:Binding affinity against Adenosine A2a receptor from rat brain tissue was determined using [3H]-ZM-241,385 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec Inc

Curated by ChEMBL
LigandPNGBDBM50152243(2-Furan-2-yl-N*5*-methyl-N*5*-[2-(4-phenyl-piperaz...)
Affinity DataKi:  11nMAssay Description:Binding affinity against Adenosine A2a receptor determined using [3H]-ZM-241,385 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec Inc

Curated by ChEMBL
LigandPNGBDBM50163403(CHEMBL368070 | N*5*-[(R)-1-(2,4-Dichloro-benzyl)-p...)
Affinity DataKi:  11nMAssay Description:Inhibition of [3H]ZM-241385 binding to adenosine A2a receptor of rat brain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec Inc

Curated by ChEMBL
LigandPNGBDBM50151205(5-[4-(2-Chloro-6-methyl-quinolin-3-ylmethyl)-piper...)
Affinity DataKi:  12nMAssay Description:Inhibition of [3H]-ZM-241,385 binidng to rat brain adenosine A2a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec Inc

Curated by ChEMBL
LigandPNGBDBM50163426(CHEMBL177539 | N*5*-((R)-1-Benzofuran-2-ylmethyl-p...)
Affinity DataKi:  12nMAssay Description:Inhibition of [3H]ZM-241385 binding to adenosine A2a receptor of rat brain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec Inc

Curated by ChEMBL
LigandPNGBDBM50152213(2-Furan-2-yl-N*5*-methyl-N*5*-[(R)-1-(5-methyl-iso...)
Affinity DataKi:  12nMAssay Description:Inhibition of [3H]ZM-241385 binding to adenosine A2a receptor of rat brain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec Inc

Curated by ChEMBL
LigandPNGBDBM50152213(2-Furan-2-yl-N*5*-methyl-N*5*-[(R)-1-(5-methyl-iso...)
Affinity DataKi:  12nMAssay Description:Binding affinity against Adenosine A2a receptor from rat brain tissue was determined using [3H]-ZM-241,385 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec Inc

Curated by ChEMBL
LigandPNGBDBM50163399(CHEMBL177943 | N*5*-[(R)-1-(2,4-Difluoro-benzyl)-p...)
Affinity DataKi:  14nMAssay Description:Inhibition of [3H]ZM-241385 binding to adenosine A2a receptor of rat brain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec Inc

Curated by ChEMBL
LigandPNGBDBM50163398(CHEMBL175645 | N*5*-[(R)-1-(3-Chloro-benzyl)-pyrro...)
Affinity DataKi:  14nMAssay Description:Inhibition of [3H]ZM-241385 binding to adenosine A2a receptor of rat brain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec Inc

Curated by ChEMBL
LigandPNGBDBM50151188(5-(4-((5-chloro-1-methyl-3-(trifluoromethyl)-1H-py...)
Affinity DataKi:  14nMAssay Description:Inhibition of [3H]-ZM-241,385 binidng to rat brain adenosine A2a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec Inc

Curated by ChEMBL
LigandPNGBDBM50163415(2-Furan-2-yl-N*5*-methyl-N*5*-[(R)-1-(5-methyl-iso...)
Affinity DataKi:  14nMAssay Description:Inhibition of [3H]ZM-241385 binding to adenosine A2a receptor of rat brain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec Inc

Curated by ChEMBL
LigandPNGBDBM50163416(2-Furan-2-yl-N*5*-((R)-1-pyridin-2-ylmethyl-pyrrol...)
Affinity DataKi:  15nMAssay Description:Inhibition of [3H]ZM-241385 binding to adenosine A2a receptor of rat brain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec Inc

Curated by ChEMBL
LigandPNGBDBM50151198(5-[4-(2,6-Difluoro-benzyl)-piperazin-1-yl]-2-furan...)
Affinity DataKi:  16nMAssay Description:Inhibition of [3H]-ZM-241,385 binidng to rat brain adenosine A2a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec Inc

Curated by ChEMBL
LigandPNGBDBM50163406(2-Furan-2-yl-N*5*-((R)-1-quinolin-2-ylmethyl-pyrro...)
Affinity DataKi:  17nMAssay Description:Inhibition of [3H]ZM-241385 binding to adenosine A2a receptor of rat brain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec Inc

Curated by ChEMBL
LigandPNGBDBM50152207(CHEMBL435099 | N*5*-[(R)-1-(2,6-Dichloro-benzyl)-p...)
Affinity DataKi:  18nMAssay Description:Binding affinity against Adenosine A2a receptor from rat brain tissue was determined using [3H]-ZM-241,385 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec Inc

Curated by ChEMBL
LigandPNGBDBM50151208(2-Furan-2-yl-5-[4-(2,3,6-trichloro-benzyl)-piperaz...)
Affinity DataKi:  18nMAssay Description:Inhibition of [3H]-ZM-241,385 binidng to rat brain adenosine A2a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec Inc

Curated by ChEMBL
LigandPNGBDBM50151195(5-[4-(3,5-Dimethyl-isoxazol-4-ylmethyl)-piperazin-...)
Affinity DataKi:  18nMAssay Description:Inhibition of [3H]-ZM-241,385 binidng to rat brain adenosine A2a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec Inc

Curated by ChEMBL
LigandPNGBDBM50151195(5-[4-(3,5-Dimethyl-isoxazol-4-ylmethyl)-piperazin-...)
Affinity DataKi:  18nMAssay Description:Inhibition of [3H]ZM-241385 binding to adenosine A2a receptor of rat brain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec Inc

Curated by ChEMBL
LigandPNGBDBM50163417(2-Furan-2-yl-N*5*-((R)-1-furan-2-ylmethyl-pyrrolid...)
Affinity DataKi:  18nMAssay Description:Inhibition of [3H]ZM-241385 binding to adenosine A2a receptor of rat brain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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