Affinity DataIC50: 500nMAssay Description:Inhibition of dopamine receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+3nMAssay Description:Antagonist activity at alpha 1a adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+3nMAssay Description:Agonist activity at 5HT1A receptor (unknown origin)More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Genentech
Curated by ChEMBL
Genentech
Curated by ChEMBL
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of human ERG expressed in HEK293 cells after 5 mins by patch clamp assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.90E+3nMAssay Description:Antagonist activity at 5HT1A receptor (unknown origin)More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase kinase 4(Homo sapiens (Human))
Genentech
Curated by ChEMBL
Genentech
Curated by ChEMBL
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibition of MAP4K4 (unknown origin) by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.30E+3nMAssay Description:Reversible inhibition of CYP3A4 (unknown origin) using testosterone as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 7.50E+3nMAssay Description:Reversible inhibition of CYP3A4 (unknown origin) using midazolam as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 2.30E+4nMAssay Description:Inhibition of GSK3beta in human human MM1S cellsMore data for this Ligand-Target Pair