Compile Data Set for Download or QSAR
maximum 50k data
Found 9 of ic50 for monomerid = 150275
TargetMineralocorticoid receptor(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM150275(US8987239, A | US9034856, A)
Affinity DataIC50:  3.30nMAssay Description:Using cytosol from progesterone receptor-expressing insect cells (Hi5), competitive binding to the progesterone receptor was determined from the abil...More data for this Ligand-Target Pair
In DepthDetails US PatentDrugBank

TargetAndrogen receptor(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM150275(US8987239, A | US9034856, A)
Affinity DataIC50:  27nMAssay Description:Using cytosol from progesterone receptor-expressing insect cells (Hi5), competitive binding to the progesterone receptor was determined from the abil...More data for this Ligand-Target Pair
In DepthDetails US PatentDrugBank

TargetProgesterone receptor(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM150275(US8987239, A | US9034856, A)
Affinity DataIC50:  43.3nMAssay Description:Using cytosol from progesterone receptor-expressing insect cells (Hi5), competitive binding to the progesterone receptor was determined from the abil...More data for this Ligand-Target Pair
In DepthDetails US PatentDrugBank

TargetProgesterone receptor(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM150275(US8987239, A | US9034856, A)
Affinity DataIC50:  43.3nMAssay Description:Using cytosol from progesterone receptor-expressing insect cells (Hi5), competitive binding to the progesterone receptor was determined from the abil...More data for this Ligand-Target Pair
In DepthDetails US PatentDrugBank

TargetAndrogen receptor(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM150275(US8987239, A | US9034856, A)
Affinity DataIC50:  630nMAssay Description:The test was carried out as in 1, with the following modifications: cytosol from androgen receptor-expressing insect cells (Hi5) was used, and the re...More data for this Ligand-Target Pair
In DepthDetails US PatentDrugBank

TargetAndrogen receptor(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM150275(US8987239, A | US9034856, A)
Affinity DataIC50:  630nMAssay Description:Using cytosol from progesterone receptor-expressing insect cells (Hi5), competitive binding to the progesterone receptor was determined from the abil...More data for this Ligand-Target Pair
In DepthDetails US PatentDrugBank

TargetBile salt export pump(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM150275(US8987239, A | US9034856, A)
Affinity DataIC50:  1.64E+4nMAssay Description:Inhibition of human BSEP overexpressed in Sf9 cell membrane vesicles assessed as uptake of [3H]-taurocholate in presence of ATP measured after 15 to ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 4(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM150275(US8987239, A | US9034856, A)
Affinity DataIC50:  3.79E+4nMAssay Description:Inhibition of human MRP4 overexpressed in Sf9 cell membrane vesicles assessed as uptake of [3H]-estradiol-17beta-D-glucuronide in presence of ATP and...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-binding cassette sub-family C member 3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM150275(US8987239, A | US9034856, A)
Affinity DataIC50: >1.33E+5nMAssay Description:Inhibition of human MRP3 overexpressed in Sf9 insect cell membrane vesicles assessed as uptake of [3H]-estradiol-17beta-D-glucuronide in presence of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed