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Found 9 of ic50 for monomerid = 154576
TargetCyclin-dependent kinase 8(Homo sapiens (Human))
Hefei University Of Technology

Curated by ChEMBL
LigandPNGBDBM154576(K03861 (1))
Affinity DataIC50:  3nMAssay Description:Inhibition of NanoLuc-fused CDK8 (unknown origin) expressed in human HEK293 cells using NanoGlo substrate incubated for 2 hrs by NanoBRET assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-dependent kinase 2 [C118L,A144C](Homo sapiens (Human))
University of Oxford

LigandPNGBDBM154576(K03861 (1))
Affinity DataIC50:  800nMpH: 7.5Assay Description:For IC50 measurements, a 384-well microtiter plate contained 8-point serial dilutions of inhibitors and 16-point serial dilutions of staurosporine as...More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2 [C118L](Homo sapiens (Human))
University of Oxford

LigandPNGBDBM154576(K03861 (1))
Affinity DataIC50:  7.20E+3nMpH: 7.5Assay Description:For IC50 measurements, a 384-well microtiter plate contained 8-point serial dilutions of inhibitors and 16-point serial dilutions of staurosporine as...More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2 [A144C](Homo sapiens (Human))
University of Oxford

LigandPNGBDBM154576(K03861 (1))
Affinity DataIC50: >1.00E+4nMpH: 7.5Assay Description:For IC50 measurements, a 384-well microtiter plate contained 8-point serial dilutions of inhibitors and 16-point serial dilutions of staurosporine as...More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2 [A144G](Homo sapiens (Human))
University of Oxford

LigandPNGBDBM154576(K03861 (1))
Affinity DataIC50: >1.00E+4nMpH: 7.5Assay Description:For IC50 measurements, a 384-well microtiter plate contained 8-point serial dilutions of inhibitors and 16-point serial dilutions of staurosporine as...More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2 [F80M](Homo sapiens (Human))
University of Oxford

LigandPNGBDBM154576(K03861 (1))
Affinity DataIC50: >1.00E+4nMpH: 7.5Assay Description:For IC50 measurements, a 384-well microtiter plate contained 8-point serial dilutions of inhibitors and 16-point serial dilutions of staurosporine as...More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2 [F80T](Homo sapiens (Human))
University of Oxford

LigandPNGBDBM154576(K03861 (1))
Affinity DataIC50: >1.00E+4nMpH: 7.5Assay Description:For IC50 measurements, a 384-well microtiter plate contained 8-point serial dilutions of inhibitors and 16-point serial dilutions of staurosporine as...More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
University of Oxford

LigandPNGBDBM154576(K03861 (1))
Affinity DataIC50: >1.00E+4nMpH: 7.5Assay Description:For IC50 measurements, a 384-well microtiter plate contained 8-point serial dilutions of inhibitors and 16-point serial dilutions of staurosporine as...More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2 [C118I](Homo sapiens (Human))
University of Oxford

LigandPNGBDBM154576(K03861 (1))
Affinity DataIC50: >1.00E+4nMpH: 7.5Assay Description:For IC50 measurements, a 384-well microtiter plate contained 8-point serial dilutions of inhibitors and 16-point serial dilutions of staurosporine as...More data for this Ligand-Target Pair