Affinity DataKi: 19nMAssay Description:Inhibition of human kidney SGLT2 assessed as renal glucose reabsorptionMore data for this Ligand-Target Pair
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Max-Planck-Institut F£R Molekulare Physiologie
Curated by ChEMBL
Max-Planck-Institut F£R Molekulare Physiologie
Curated by ChEMBL
Affinity DataKi: 180nMAssay Description:Binding affinity against Sodium/glucose co-transporter of isolated renal brush border membranes.More data for this Ligand-Target Pair
TargetSolute carrier family 28 member 3(Homo sapiens (Human))
University Of Tennessee Health Sciences Center
Curated by ChEMBL
University Of Tennessee Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 1.60E+4nMAssay Description:Binding affinity to human recombinant CNT3 expressed in pig PK15NTD cells assessed as [3H]uridine uptake by beta-scintillation counterMore data for this Ligand-Target Pair
Affinity DataKi: 6.43E+4nMAssay Description:Inhibition of diphenolase activity of mushroom tyrosinaseMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University Of Tennessee Health Sciences Center
Curated by ChEMBL
University Of Tennessee Health Sciences Center
Curated by ChEMBL
Affinity DataKi: >1.00E+6nMAssay Description:Binding affinity to human ENT1 assessed as [3H]uridine uptake by flow cytometryMore data for this Ligand-Target Pair