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Found 2 of ki for monomerid = 24941
TargetSerine/threonine-protein kinase PLK3(Homo sapiens (Human))
Paradigm Pharmaceuticals

LigandPNGBDBM24941((2Z)-2-{[(2,5-dibromophenyl)amino](hydroxy)methyli...)
Affinity DataKi:  7.20E+3nM ΔG°:  -6.94kcal/mole IC50:  6.10E+4nMpH: 7.0 T: 2°CAssay Description:The mode of human PLK3 inhibition by LFM-A13 was examined in titration experiments using increasing concentrations of [gamma-32P]ATP and purified N-t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHomoserine kinase(Escherichia coli)
Mcmaster University

LigandPNGBDBM24941((2Z)-2-{[(2,5-dibromophenyl)amino](hydroxy)methyli...)
Affinity DataKi:  1.20E+4nM ΔG°:  -6.98kcal/molepH: 7.5 T: 2°CAssay Description:The phosphorylation of L-Hse was monitored by coupling the formation of ADP with pyruvate kinase and lactate dehydrogenase (PK/LDH). The resulting o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed