Compile Data Set for Download or QSAR
maximum 50k data
Found 8 of ec50 for monomerid = 36894
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM36894(5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide ...)
Affinity DataEC50:  3.22E+3nMAssay Description:Source (MLSCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute, TSRI Assay ...More data for this Ligand-Target Pair
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TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM36894(5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide ...)
Affinity DataEC50: >9.51E+4nMAssay Description:Source (MLSCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute, TSRI Assay ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM36894(5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide ...)
Affinity DataEC50:  3.95E+3nMAssay Description:Source (MLSCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute, TSRI Assay ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Columbia University

Curated by ChEMBL
LigandPNGBDBM36894(5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide ...)
Affinity DataEC50:  2.60E+3nMAssay Description:Induction of human IkappaBalpha stabilization in OCI-Ly3 cells assessed as ratio of green light emiting IkappaBalpha-fused luciferase expression to r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4(Homo sapiens (Human))
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM36894(5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide ...)
Affinity DataEC50:  1.99E+4nMAssay Description:Assay Support: 1 X01 MH077638-01 MLSCN Assay for Allosteric Ligands for the VLA-4 Integrin PI: SKLAR, LARRY A University of New Mexico Assay Overview...More data for this Ligand-Target Pair
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TargetHeat shock factor protein 1(Mus musculus)
Broad Institute

Curated by PubChem BioAssay
LigandPNGBDBM36894(5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide ...)
Affinity DataEC50:  2.76E+3nMAssay Description:Keywords: Heat Shock Factor-1 (HSF-1), Stress Response, MG132, NIH3T3, Luminescence Assay Overview: Confirmation testing of small molecules identifie...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Columbia University

Curated by ChEMBL
LigandPNGBDBM36894(5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide ...)
Affinity DataEC50:  2.20E+3nMAssay Description:Induction of human IkappaBalpha stabilization in OCI-Ly3 cells by green light emiting IkappaBalpha-fused luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-14 [1-36](Homo sapiens (Human))
Sanford-Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM36894(5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide ...)
Affinity DataEC50:  2.46E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay