TargetSigma non-opioid intracellular receptor 1(RAT)
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of [3H]NANM binding to sigma receptor obtained from tissue homogenate preparation of fresh whole rat brain minus cerebellumMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(RAT)
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:In vitro for binding affinity against sigma receptor using [3H](+)-3-PPP as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 98nMAssay Description:In vitro inhibition of [3H]-N-0437 binding to Dopamine receptor D2 in rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 230nMAssay Description:Displacement of spiperone from dopamine receptor D2 of rat brain membraneChecked by AuthorMore data for this Ligand-Target Pair
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rattus norvegicus (rat))
Warner-Lambert
Curated by ChEMBL
Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 930nMAssay Description:In vitro inhibition of [3H]haloperidol (HPD) binding to dopamine (DA) receptor of rat striatal membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(RAT)
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
Affinity DataIC50: 1.52E+3nMAssay Description:Displacement of (+)-3PPP from sigma receptor of rat brain membraneChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.71E+3nMAssay Description:Binding affinity against Dopamine receptor D2 using [3H]spiperone as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 2.30E+4nMAssay Description:In vitro inhibition of [3H]-spiperone binding to Dopamine receptor D2 in rat striatal membranesMore data for this Ligand-Target Pair
TargetLysosomal Pro-X carboxypeptidase(Homo sapiens (Human))
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of binding to PCP receptor obtained from tissue homogenate preparation of fresh whole rat brain minus cerebellumMore data for this Ligand-Target Pair