TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
Moltech
Curated by ChEMBL
Moltech
Curated by ChEMBL
Affinity DataEC50: 7.44E+4nMAssay Description:Activity at GABAA alpha-1-beta-3-gamma-2 receptor expressed in Xenopus oocytes assessed as inhibition of GABA-induced current by voltage clamp assayMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-2(Homo sapiens (Human))
Moltech
Curated by ChEMBL
Moltech
Curated by ChEMBL
Affinity DataEC50: 9.55E+4nMAssay Description:Activity at alpha-2-beta-3-gamma-2 GABAA receptor expressed in Xenopus oocytes assessed as inhibition in GABA-induced current by voltage clamp assayMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-6(Homo sapiens (Human))
Moltech
Curated by ChEMBL
Moltech
Curated by ChEMBL
Affinity DataEC50: 5.17E+4nMAssay Description:Activity at alpha-6-beta-3-gamma-2 GABAA receptor expressed in Xenopus oocytes assessed as inhibition in GABA-induced current by voltage clamp assayMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-5(Homo sapiens (Human))
Moltech
Curated by ChEMBL
Moltech
Curated by ChEMBL
Affinity DataEC50: 9.80E+3nMAssay Description:Activity at alpha-5-beta-3-gamma-2 GABAA receptor expressed in Xenopus oocytes assessed as inhibition in GABA-induced current by voltage clamp assayMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-4(Homo sapiens (Human))
Moltech
Curated by ChEMBL
Moltech
Curated by ChEMBL
Affinity DataEC50: 3.24E+5nMAssay Description:Activity at alpha-4-beta-3-gamma-2 GABAA receptor expressed in Xenopus oocytes assessed as inhibition in GABA-induced current by voltage clamp assayMore data for this Ligand-Target Pair