Compile Data Set for Download or QSAR
maximum 50k data
Found 17 of ki for monomerid = 50055520
TargetD(3) dopamine receptor(Homo sapiens (Human))
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50055520(CHEMBL3321789)
Affinity DataKi:  4.10nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D3 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50055520(CHEMBL3321789)
Affinity DataKi:  20nMAssay Description:Displacement [3H]-DTG from sigma 2 receptor (unknown origin) expressed in HEK cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50055520(CHEMBL3321789)
Affinity DataKi:  20nMAssay Description:Displacement [3H]-DTG from sigma 2 receptor (unknown origin) expressed in HEK cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50055520(CHEMBL3321789)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D2 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(RAT)
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50055520(CHEMBL3321789)
Affinity DataKi:  49nMAssay Description:Displacement of [3H]N-methylspiperone from rat dopamine D4 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50055520(CHEMBL3321789)
Affinity DataKi:  123nMAssay Description:Displacement of [3H] 8-OH-DPAT from human 5-HT1A receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50055520(CHEMBL3321789)
Affinity DataKi:  166nMAssay Description:Displacement [3H]-Pentazocine from sigma 1 receptor (unknown origin) expressed in HEK cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50055520(CHEMBL3321789)
Affinity DataKi:  166nMAssay Description:Displacement [3H]-Pentazocine from sigma 1 receptor (unknown origin) expressed in HEK cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50055520(CHEMBL3321789)
Affinity DataKi:  236nMAssay Description:Displacement of [3H]Ketanserin from human 5-HT2A receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50055520(CHEMBL3321789)
Affinity DataKi:  255nMAssay Description:Displacement of [3H]Citalopram from human Serotonin transporter by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50055520(CHEMBL3321789)
Affinity DataKi:  420nMAssay Description:Displacement of [3H]LSD from human 5-HT7 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50055520(CHEMBL3321789)
Affinity DataKi:  620nMAssay Description:Displacement of [3H]GBR12935 from human dopamine transporter by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50055520(CHEMBL3321789)
Affinity DataKi:  898nMAssay Description:Displacement of [3H]LSD from human 5-HT2B receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50055520(CHEMBL3321789)
Affinity DataKi:  1.79E+3nMAssay Description:Displacement of [3H]Nisoxetine from human Norepinephrine transporter by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50055520(CHEMBL3321789)
Affinity DataKi:  4.15E+3nMAssay Description:Displacement of [3H]Pyrilamine from human histamine H1 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50055520(CHEMBL3321789)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D5 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50055520(CHEMBL3321789)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D1 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed