TargetD(3) dopamine receptor(Homo sapiens (Human))
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Affinity DataKi: 0.100nMAssay Description:Displacement of [3H]methylspiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Displacement of [3H]LSD from human recombinant 5-HT6 receptor expressed in HEK-293 cells incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Affinity DataKi: 6.30nMAssay Description:Displacement of [3H]methylspiperone from human D2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Affinity DataKi: 6.30nMAssay Description:Displacement of [3H]N-methylspiperone from human recombinant dopamine D2 receptor expressed in CHOK1 cells incubated for 60 mins by scintillation cou...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Affinity DataKi: 6.70nMAssay Description:Displacement of [3H]-8-OH-DPAT from human 5-HT1A receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
TargetD(4) dopamine receptor(Homo sapiens (Human))
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Affinity DataKi: 7.10nMAssay Description:Displacement of [3H]methylspiperone from human dopamine D4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Displacement of [3H]prazosin from human adrenergic alpha1A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Affinity DataKi: 29nMAssay Description:Displacement of [3H]ketanserin from human 5-HT2A receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Affinity DataKi: 160nMAssay Description:Displacement of [3H]pyrilamine from human histamine H1 receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Affinity DataKi: 180nMAssay Description:Displacement of [3H]LSD from human 5-HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Affinity DataKi: 190nMAssay Description:Displacement of [3H]RX-821002 from human adrenergic alpha2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]pirenzepine from human muscarinic M1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]imipramine from human SERT expressed in CHO cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]mesulergine from human 5-HT2C receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair